SCHEMBL6869841

SCHEMBL6869841

CCN(Cc1ccccc1F)C(=O)c1cc(N)n2nc(-c3cccnc3)nc2c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 5/20 0.48
ADRB2 P07550 1/20 0.41
HSD17B10 Q99714 2/20 0.40
KDM4E B2RXH2 1/20 0.40
F2 P00734 4/20 0.40
KMT2A Q03164 3/20 0.40
CYP1A2 P05177 1/20 0.40
HPGD P15428 1/20 0.40
CYP2C19 P33261 1/20 0.40
MAPT P10636 2/20 0.38
F12 P00748 1/20 0.38
RAB9A P51151 1/20 0.37
TSPO P30536 1/20 0.37
KLK7 P49862 1/20 0.36
KLK14 Q9P0G3 1/20 0.36
KLK5 Q9Y337 1/20 0.36
ST14 Q9Y5Y6 1/20 0.36
NPY2R P49146 1/20 0.36
ALDH1A1 P00352 1/20 0.35
HTT P42858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6871681 0.88 ADORA2A (0.51) ADORA2AHSD17B10KDM4EF2KMT2A
SCHEMBL6867466 0.82 ADORA2A (0.49) ADORA2AHSD17B10KDM4EHPGDTSPO
SCHEMBL6868330 0.79 ADORA2A (0.45) ADORA2AHSD17B10F2KMT2ACYP1A2
SCHEMBL6870143 0.79 ADORA2A (0.65) ADORA2AKDM4EKMT2AHPGDMAPT
SCHEMBL6863381 0.79 ADORA2A (0.46) ADORA2AHSD17B10KDM4EHPGDMAPT
SCHEMBL6872977 0.78 ADORA2A (0.51) ADORA2AHSD17B10KDM4EF2KMT2A
SCHEMBL6866915 0.77 PSMB5 (0.51) ADORA2AHSD17B10KDM4EF2KMT2A
SCHEMBL6871922 0.73 CYP19A1 (0.54) HSD17B10KDM4EF2KMT2ACYP1A2
SCHEMBL6863310 0.72 ADORA2A (0.64) ADORA2AHSD17B10F2HPGDF12
SCHEMBL6871512 0.72 KMT2A (0.49) ADORA2AHSD17B10F2KMT2ACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed