SCHEMBL6871922

SCHEMBL6871922

COC(=O)c1cc(N)n2nc(-c3cccnc3)nc2c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.54
CYP11B1 P15538 1/20 0.54
CYP11B2 P19099 1/20 0.54
F12 P00748 5/20 0.47
KLK3 P07288 3/20 0.47
EGFR P00533 1/20 0.47
TUBB4A P04350 1/20 0.47
TUBB P07437 1/20 0.47
TUBA3C P0DPH7 1/20 0.47
TUBA1B P68363 1/20 0.47
TUBA4A P68366 1/20 0.47
TUBB4B P68371 1/20 0.47
TUBB3 Q13509 1/20 0.47
TUBB2A Q13885 1/20 0.47
TUBB8 Q3ZCM7 1/20 0.47
TUBA3E Q6PEY2 1/20 0.47
TUBA1A Q71U36 1/20 0.47
TUBA1C Q9BQE3 1/20 0.47
TUBB6 Q9BUF5 1/20 0.47
TUBB2B Q9BVA1 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6871212 0.87 ALDH1A1 (0.48) ALDH1A1MAPTKMT2AKLK7KLK5
SCHEMBL6867215 0.80 PLAU (0.47) EGFRF2POLBKMT2ACYP1A2
SCHEMBL6869675 0.80 ALDH1A1 (0.54) F12KLK3ALDH1A1F2POLB
SCHEMBL6867024 0.80 F12 (0.41) F12KLK3F2MAPTKMT2A
SCHEMBL6867019 0.79 DYRK1A (0.47) F12ALDH1A1ABL1KDM4E
SCHEMBL6867379 0.78 ADORA2A (0.66) F12KLK3F2KDM4E
SCHEMBL6871806 0.78 ADORA2A (0.42)
SCHEMBL6872919 0.77 KDM4A (0.52) ALDH1A1POLBMAPTKMT2AHPGD
SCHEMBL6871512 0.77 KMT2A (0.49) F12ALDH1A1F2MAPTKMT2A
SCHEMBL6871681 0.76 ADORA2A (0.51) F12ALDH1A1F2MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed