SCHEMBL6870449

SCHEMBL6870449

Cc1ccc(-c2nc3cc(C(=O)Nc4ccccc4)cc(N)n3n2)s1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 6/20 0.45
NPC1 O15118 5/20 0.45
ADORA2A P29274 3/20 0.44
TP53 P04637 1/20 0.43
ALDH1A1 P00352 3/20 0.42
LMNA P02545 1/20 0.42
RECQL P46063 1/20 0.42
PDE5A O76074 1/20 0.41
PDE1A P54750 1/20 0.41
PDE1B Q01064 1/20 0.41
PDE1C Q14123 1/20 0.41
HDAC3 O15379 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC2 Q92769 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
MAPT P10636 2/20 0.41
IKBKE Q14164 1/20 0.41
TBK1 Q9UHD2 1/20 0.41
MEN1 O00255 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6869624 0.88 ADORA2A (0.41) RAB9ANPC1ADORA2ATP53ALDH1A1
SCHEMBL6863351 0.85 PLAU (0.47) ADORA2ATP53ALDH1A1LMNAHDAC3
SCHEMBL6871437 0.84 ADORA2A (0.47) RAB9ANPC1ADORA2AALDH1A1HTT
SCHEMBL6863751 0.84 ADORA2A (0.62) RAB9ANPC1ADORA2ATP53ALDH1A1
SCHEMBL6868100 0.83 ADORA2A (0.44) RAB9ANPC1ADORA2ATP53ALDH1A1
SCHEMBL6870464 0.81 ADORA2A (0.42) RAB9ANPC1ADORA2AALDH1A1LMNA
SCHEMBL6868343 0.81 ADORA2A (0.45) RAB9ANPC1ADORA2AALDH1A1MAPT
SCHEMBL6867554 0.80 ADORA2A (0.63) ADORA2AALDH1A1HDAC1MAPTMEN1
SCHEMBL6867499 0.79 KMT2A (0.43) ADORA2AALDH1A1LMNAHDAC3HDAC1
SCHEMBL6870466 0.79 TP53 (0.47) TP53ALDH1A1LMNAMAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed