SCHEMBL6868100

SCHEMBL6868100

Nc1cc(C(=O)Nc2ccccc2)cc2nc(-c3ccccc3)nn12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 3/20 0.44
PTPN1 P18031 1/20 0.43
PLAU P00749 1/20 0.43
ALOX5 P09917 1/20 0.43
ALDH1A1 P00352 4/20 0.43
RAB9A P51151 4/20 0.43
LMNA P02545 3/20 0.43
NPC1 O15118 3/20 0.43
MAPT P10636 3/20 0.42
TP53 P04637 1/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
SMN1; SMN2 Q16637 4/20 0.42
HPGD P15428 3/20 0.42
NFKB1 P19838 1/20 0.42
HTT P42858 1/20 0.42
NFKB2 Q00653 1/20 0.42
RELA Q04206 1/20 0.42
POLB P06746 2/20 0.42
GAA P10253 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6869842 0.88 PLAU (0.48) ADORA2APLAUALOX5ALDH1A1RAB9A
SCHEMBL6868483 0.85 ADORA2A (0.64) ADORA2APLAU
SCHEMBL6870681 0.84 ADORA2A (0.49) ADORA2AALDH1A1RAB9ANPC1MAPT
SCHEMBL6863751 0.84 ADORA2A (0.62) ADORA2AALDH1A1RAB9ALMNANPC1
SCHEMBL6868263 0.83 MAPT (0.46) ADORA2APLAUALOX5ALDH1A1RAB9A
SCHEMBL6870449 0.83 RAB9A (0.45) ADORA2APLAUALDH1A1RAB9ALMNA
SCHEMBL6869736 0.82 ADORA2A (0.48) ADORA2A
SCHEMBL6873045 0.82 ADORA2A (0.62) ADORA2AMAPTMEN1KMT2ASMN1; SMN2
SCHEMBL6871948 0.82 HDAC2 (0.46) ADORA2AALDH1A1RAB9ALMNANPC1
SCHEMBL6867554 0.82 ADORA2A (0.63) ADORA2AALDH1A1MAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed