SCHEMBL6863751

SCHEMBL6863751

Nc1cc(C(=O)Nc2ccccc2)cc2nc(-c3cccs3)nn12

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 2/20 0.62
ALDH1A1 P00352 5/20 0.46
MAPT P10636 3/20 0.46
GAA P10253 2/20 0.46
HTT P42858 2/20 0.46
ALOX15 P16050 1/20 0.46
MAPK1 P28482 1/20 0.46
HSD17B10 Q99714 1/20 0.46
GRM5 P41594 1/20 0.46
HDAC3 O15379 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC2 Q92769 1/20 0.42
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
MEN1 O00255 5/20 0.41
KMT2A Q03164 5/20 0.41
HPGD P15428 3/20 0.41
NPSR1 Q6W5P4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7153750 0.85 ADORA2A (0.71) ADORA2AALDH1A1HTTKDM4EADORA3
SCHEMBL6868100 0.84 ADORA2A (0.44) ADORA2AALDH1A1MAPTGAAHTT
SCHEMBL6870449 0.84 RAB9A (0.45) ADORA2AALDH1A1MAPTHTTHDAC3
SCHEMBL6871948 0.83 HDAC2 (0.46) ADORA2AALDH1A1HTTHDAC3HDAC1
SCHEMBL6870464 0.82 ADORA2A (0.42) ADORA2AALDH1A1MAPTGRM5HDAC1
SCHEMBL6870583 0.81 ADORA2A (0.66) ADORA2AALDH1A1MAPTGAAHSD17B10
SCHEMBL6869624 0.81 ADORA2A (0.41) ADORA2AALDH1A1MAPTHTTALOX15
SCHEMBL6863748 0.79 ADORA2A (0.64) ADORA2AALDH1A1MAPTHTTHSD17B10
SCHEMBL6870384 0.79 ADORA2A (0.58) ADORA2AALDH1A1MAPTGAAHTT
SCHEMBL6868483 0.79 ADORA2A (0.64) ADORA2ACYP3A4CYP2C9KCNK3KCNK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed