SCHEMBL6872186

SCHEMBL6872186

CCCCNC(=O)c1cc(N)n2nc(-c3ccccc3O)nc2c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.43
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
HPGD P15428 1/20 0.41
CYP2C19 P33261 1/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
NAAA Q02083 2/20 0.40
TSHR P16473 2/20 0.40
HTT P42858 1/20 0.40
ADORA2A P29274 3/20 0.39
EGLN2 Q96KS0 1/20 0.39
BACE1 P56817 1/20 0.39
TP53 P04637 2/20 0.39
LMNA P02545 1/20 0.39
KDR P35968 1/20 0.39
BCL2 P10415 1/20 0.39
MCL1 Q07820 1/20 0.39
RXFP1 Q9HBX9 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6866973 0.86 BACE1 (0.48) SMN1; SMN2HPGDNPC1RAB9ANAAA
SCHEMBL6869989 0.83 ADORA2A (0.58) SMN1; SMN2NPC1RAB9ANAAAHTT
SCHEMBL6871320 0.81 SMN1; SMN2 (0.43) SMN1; SMN2HPGDNPC1RAB9ANAAA
SCHEMBL6870605 0.81 ADORA2A (0.58) HPGDADORA2AMCL1
SCHEMBL6870384 0.81 ADORA2A (0.58) SMN1; SMN2HPGDHTTADORA2AEGLN2
SCHEMBL6867215 0.80 PLAU (0.47) SMN1; SMN2CYP1A2HPGDCYP2C19TP53
SCHEMBL6869214 0.80 KMT2A (0.46) ADORA2ALMNA
SCHEMBL6868276 0.80 TP53 (0.44) SMN1; SMN2CYP1A2CYP3A4HPGDCYP2C19
SCHEMBL6871700 0.80 SMN1; SMN2 (0.41) SMN1; SMN2HPGDNPC1RAB9AADORA2A
SCHEMBL6872919 0.79 KDM4A (0.52) SMN1; SMN2HPGDADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed