SCHEMBL6866973

SCHEMBL6866973

CCCCNC(=O)c1cc(N)n2nc(-c3ccccc3)nc2c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.48
ALOX15 P16050 4/20 0.47
SMN1; SMN2 Q16637 3/20 0.46
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
POLB P06746 2/20 0.46
KDM4E B2RXH2 2/20 0.46
ALDH1A1 P00352 2/20 0.46
TP53 P04637 2/20 0.46
HTT P42858 2/20 0.46
HCRTR1 O43613 1/20 0.46
NAAA Q02083 1/20 0.45
EGLN2 Q96KS0 1/20 0.43
DRD2 P14416 1/20 0.43
DRD4 P21917 1/20 0.43
DRD3 P35462 1/20 0.43
MAPT P10636 1/20 0.43
HPGD P15428 2/20 0.42
GAA P10253 1/20 0.42
CAMK2D Q13557 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6867215 0.89 PLAU (0.47) SMN1; SMN2POLBTP53HPGDCAMK2D
SCHEMBL6872186 0.86 SMN1; SMN2 (0.43) BACE1SMN1; SMN2NPC1RAB9ATP53
SCHEMBL6869989 0.85 ADORA2A (0.58) SMN1; SMN2NPC1RAB9AHTTNAAA
SCHEMBL6870530 0.85 ADORA2A (0.43) BACE1ALOX15SMN1; SMN2NPC1RAB9A
SCHEMBL6870384 0.83 ADORA2A (0.58) BACE1ALOX15SMN1; SMN2KDM4EALDH1A1
SCHEMBL6870605 0.83 ADORA2A (0.58) ALOX15POLBKDM4EALDH1A1MAPT
SCHEMBL6871320 0.83 SMN1; SMN2 (0.43) BACE1ALOX15SMN1; SMN2NPC1RAB9A
SCHEMBL6873157 0.83 HPGDS (0.51) KDM4EALDH1A1HPGDTSHR
SCHEMBL6871700 0.82 SMN1; SMN2 (0.41) BACE1ALOX15SMN1; SMN2NPC1RAB9A
SCHEMBL6872486 0.82 ADORA2A (0.56) ALOX15SMN1; SMN2TP53NAAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed