SCHEMBL687314

SCHEMBL687314

CNc1n[nH]cc1-c1nc2ccccc2s1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ILK Q13418 7/20 0.56
KDM4E B2RXH2 6/20 0.51
MEN1 O00255 5/20 0.51
KMT2A Q03164 5/20 0.51
ALDH1A1 P00352 5/20 0.51
NPC1 O15118 4/20 0.51
RAB9A P51151 4/20 0.51
SMN1; SMN2 Q16637 4/20 0.51
GAA P10253 3/20 0.51
MAPT P10636 3/20 0.51
APP P05067 3/20 0.51
GLA P06280 2/20 0.51
TDP1 Q9NUW8 2/20 0.51
L3MBTL1 Q9Y468 2/20 0.51
HCRTR1 O43613 1/20 0.49
NPSR1 Q6W5P4 2/20 0.44
PKM P14618 1/20 0.44
NPY1R P25929 1/20 0.44
NPY2R P49146 1/20 0.44
POLB P06746 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10285203 0.83 GSK3B (0.58) ILKKDM4EMEN1KMT2AALDH1A1
SCHEMBL686882 0.82 ILK (0.45) ILKKDM4EMEN1KMT2AALDH1A1
SCHEMBL687432 0.81 ILK (0.56) ILKKDM4EMEN1KMT2AALDH1A1
SCHEMBL687108 0.79 KDM4E (0.61) ILKKDM4EMEN1KMT2AALDH1A1
SCHEMBL715973 0.77 ILK (0.54) ILKKDM4EMEN1KMT2AALDH1A1
SCHEMBL687313 0.74 ILK (0.56) ILKKDM4EMEN1KMT2AALDH1A1
SCHEMBL10291165 0.74 MAPT (0.63) ILKKDM4EMEN1KMT2AALDH1A1
SCHEMBL686607 0.74 ILK (0.42) ILKKDM4EMEN1KMT2AALDH1A1
SCHEMBL687376 0.73 KDM4E (0.68) KDM4EMEN1KMT2AALDH1A1NPC1
SCHEMBL686516 0.73 ALDH1A1 (0.61) ILKKDM4EMEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1542997-B1 PYRAZOLYLBENZOTHIAZOLE DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS DERMIRA CANADA INC (CA) 2012-02-29 EP disclosed