SCHEMBL6875109

SCHEMBL6875109

CN(C)c1ccnc(N[C@H]2CC[C@@H](NC(=S)NCc3cccc(Cl)c3)CC2)n1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX12 P18054 3/20 0.57
MAPT P10636 2/20 0.57
ACHE P22303 1/20 0.49
BACE1 P56817 1/20 0.49
MCHR1 Q99705 3/20 0.47
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
LMNA P02545 3/20 0.43
HTT P42858 2/20 0.43
PKM P14618 2/20 0.43
MAPK1 P28482 2/20 0.42
ADRA2A P08913 2/20 0.41
ADRA1A P35348 1/20 0.41
HRH1 P35367 1/20 0.41
HTR2B P41595 1/20 0.41
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 1/20 0.40
ALPL P05186 1/20 0.40
ALPI P09923 1/20 0.40
HPGD P15428 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6875118 1.00 ALOX12 (0.57) ALOX12MAPTACHEBACE1MCHR1
SCHEMBL6880741 0.84 ACHE (0.51) ACHEBACE1MCHR1MAPK1ADRA2A
SCHEMBL6880731 0.84 ACHE (0.51) ACHEBACE1MCHR1MAPK1ADRA2A
SCHEMBL6867794 0.83 ACHE (0.46) ALOX12MAPTACHEBACE1MCHR1
SCHEMBL6867785 0.83 ACHE (0.46) ALOX12MAPTACHEBACE1MCHR1
SCHEMBL6867777 0.82 MEN1 (0.41) MAPTACHEMCHR1RAB9ALMNA
SCHEMBL6867769 0.82 MEN1 (0.41) MAPTACHEMCHR1RAB9ALMNA
SCHEMBL4036394 0.80 MCHR1 (0.66) ALOX12MAPTMCHR1NPC1RAB9A
SCHEMBL5521361 0.80 MCHR1 (0.66) ALOX12MAPTMCHR1NPC1RAB9A
SCHEMBL7042080 0.80 ACHE (0.48) ACHEBACE1MCHR1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP disclosed