SCHEMBL6875822

SCHEMBL6875822

CN(C)c1nc(NC2CCC(NC(=S)Nc3cccc([N+](=O)[O-])c3)CC2)nc2c1CCCC2

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.54
ADRA2A P08913 1/20 0.51
MCHR1 Q99705 1/20 0.51
KMT2A Q03164 5/20 0.46
MEN1 O00255 3/20 0.46
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
ALDH1A1 P00352 3/20 0.44
CTSL P07711 2/20 0.42
CTSB P07858 2/20 0.42
CTSS P25774 2/20 0.42
CTSK P43235 2/20 0.42
POLB P06746 2/20 0.42
MAPT P10636 2/20 0.42
CCNA2 P20248 1/20 0.42
CDK2 P24941 1/20 0.42
CDK5 Q00535 1/20 0.42
CDK5R1 Q15078 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.40
LMNA P02545 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6875814 1.00 PKM (0.54) PKMADRA2AMCHR1KMT2AMEN1
SCHEMBL6877551 0.91 NPC1 (0.56) PKMADRA2AMCHR1KMT2AMEN1
SCHEMBL6877545 0.91 NPC1 (0.56) PKMADRA2AMCHR1KMT2AMEN1
SCHEMBL6875509 0.90 ALDH1A1 (0.46) PKMADRA2AMCHR1KMT2AMEN1
SCHEMBL6875517 0.90 ALDH1A1 (0.46) PKMADRA2AMCHR1KMT2AMEN1
SCHEMBL6873049 0.87 ALDH1A1 (0.45) PKMADRA2AMCHR1KMT2AMEN1
SCHEMBL6873057 0.87 ALDH1A1 (0.45) PKMADRA2AMCHR1KMT2AMEN1
SCHEMBL6871841 0.86 SMN1; SMN2 (0.55) ADRA2AMCHR1KMT2AMEN1NPC1
SCHEMBL6871842 0.86 SMN1; SMN2 (0.55) ADRA2AMCHR1KMT2AMEN1NPC1
SCHEMBL6879588 0.85 NPC1 (0.57) PKMADRA2AMCHR1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP disclosed