SCHEMBL6875901

SCHEMBL6875901

C[CH]OCc1ccc(-c2ncccn2)cc1

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 2/20 0.52
CLK4 Q9HAZ1 4/20 0.47
AOC3 Q16853 2/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
DYRK1A Q13627 1/20 0.36
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
CYP2A6 P11509 1/20 0.33
PKM P14618 1/20 0.33
DHFR P00374 1/20 0.33
IDO1 P14902 1/20 0.32
AGXT P21549 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25735768 0.79 CLK4 (0.57) ADRB2CLK4AOC3HDAC1HDAC8
SCHEMBL6878724 0.76 ADRB2 (0.62) ADRB2CLK4IDO1AGXT
SCHEMBL6875904 0.73 ADRB2 (0.53) ADRB2CLK4AOC3HDAC1HDAC8
SCHEMBL2560488 0.72 ADRB2 (0.63) ADRB2CLK4AOC3HDAC1HDAC8
SCHEMBL444754 0.72 LOXL2 (0.41)
SCHEMBL10162103 0.72 ADRB2 (0.63) ADRB2CLK4NPC1RAB9AKMT2A
SCHEMBL6854269 0.72 ADRB2 (0.49) ADRB2CLK4AOC3HDAC1HDAC8
SCHEMBL58206 0.72 TSHR (0.52) HDAC6IDO1AGXT
SCHEMBL6685962 0.71 CLK4 (0.64) ADRB2CLK4AOC3DYRK1ANPC1
SCHEMBL6853976 0.69 ADRB2 (0.59) ADRB2CLK4AOC3KMT2ACYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6825170-B2 ERYTHROMYCIN TYPE MACROLIDE WITH A FUSED OXAZOLONE RING ORTHO-MCNEIL PHARMACEUTICAL, INC. 2004-11-30 US disclosed