SCHEMBL6876444

SCHEMBL6876444

O=C(O)CCN(C1(C(=O)NO)CCCC1)S(=O)(=O)c1ccc(Oc2ccccc2)cc1

nearest known ligand 0.81

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MMP1 P03956 15/20 0.81
MMP13 P45452 13/20 0.50
MMP2 P08253 10/20 0.50
MMP9 P14780 6/20 0.50
MMP14 P50281 6/20 0.50
MMP8 P22894 5/20 0.50
MMP16 P51512 2/20 0.50
MMP3 P08254 5/20 0.48
ADAM17 P78536 1/20 0.45
LMNA P02545 1/20 0.44
ADAMTS4 O75173 2/20 0.44
ADAMTS5 Q9UNA0 2/20 0.44
MEP1B Q16820 1/20 0.43
DAGLA Q9Y4D2 1/20 0.43
PTGES O14684 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6699509 0.98 MMP1 (0.84) MMP1MMP13MMP2MMP9MMP14
SCHEMBL25130 0.92 MMP1 (0.96) MMP1MMP13MMP2MMP9MMP14
SCHEMBL6818064 0.92 MMP1 (0.78) MMP1MMP13MMP2MMP9MMP14
SCHEMBL3914710 0.92 MMP1 (0.78) MMP1MMP13MMP2MMP9MMP14
SCHEMBL6813051 0.91 MMP1 (0.94) MMP1MMP13MMP2MMP9MMP14
SCHEMBL6873149 0.91 MMP1 (0.70) MMP1MMP13MMP2MMP9MMP14
SCHEMBL26986 0.89 MMP1 (1.00) MMP1MMP13MMP2MMP9MMP14
SCHEMBL6695057 0.89 MMP1 (0.81) MMP1MMP13MMP2MMP9MMP14
SCHEMBL8502159 0.88 MMP1 (0.69) MMP1MMP13MMP2MMP9MMP14
SCHEMBL14302914 0.88 MMP1 (0.66) MMP1MMP13MMP2MMP9MMP14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6417229-B1 ENZYME INHIBITORS PFIZER INC 2002-07-09 US claimed
EP-1088550-A1 alpha-sulfonylamino hydroxamic acid inhibitors of matrix metallo-proteinases for the treatment of peripheral or central nervous system disorders Pfizer Products Inc. (US) 2001-04-04 EP claimed
EP-1415984-A1 Aryloxyarylsulfonylamino hydroxamic acid derivatives Pfizer Products Inc. (US) 2004-05-06 EP disclosed
US-6417229-B1 ENZYME INHIBITORS PFIZER INC 2002-07-09 US disclosed
US-6214872-B1 ANTIARTHRITIC AND ANTICARCINOGENIC AGENTS PFIZER INC. 2001-04-10 US disclosed
EP-1088550-A1 alpha-sulfonylamino hydroxamic acid inhibitors of matrix metallo-proteinases for the treatment of peripheral or central nervous system disorders Pfizer Products Inc. (US) 2001-04-04 EP disclosed
EP-1003720-A1 ARYLOXYARYLSULFONYLAMINO HYDROXAMIC ACID DERIVATIVES Pfizer Products Inc. (US) 2000-05-31 EP disclosed
WO-1999007675-A1 ARYLOXYARYLSULFONYLAMINO HYDROXAMIC ACID DERIVATIVES PFIZER PRODUCTS INC. (US) 1999-02-18 WO disclosed