SCHEMBL25130

SCHEMBL25130

O=C(O)CCN(C1(C(=O)NO)CCCC1)S(=O)(=O)c1ccc(Oc2ccc(F)cc2)cc1

nearest known ligand 0.96

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MMP1 P03956 17/20 0.96
MMP13 P45452 16/20 0.54
MMP9 P14780 6/20 0.47
MMP2 P08253 5/20 0.47
MMP8 P22894 4/20 0.47
MMP3 P08254 3/20 0.47
MMP14 P50281 2/20 0.47
MMP12 P39900 1/20 0.47
LTA4H P09960 1/20 0.44
FFAR1 O14842 1/20 0.41
MMP16 P51512 1/20 0.41
MEP1B Q16820 1/20 0.40
ADAM17 P78536 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6813051 0.99 MMP1 (0.94) MMP1MMP13MMP9MMP2MMP8
SCHEMBL26986 0.98 MMP1 (1.00) MMP1MMP13MMP9MMP2MMP8
SCHEMBL13556928 0.92 MMP1 (0.81) MMP1MMP13MMP9MMP2MMP8
SCHEMBL6876444 0.92 MMP1 (0.81) MMP1MMP13MMP9MMP2MMP8
SCHEMBL26434 0.91 MMP1 (0.83) MMP1MMP13MMP9MMP2MMP8
SCHEMBL4783958 0.90 MMP1 (0.79) MMP1MMP13MMP9MMP2MMP8
SCHEMBL3914710 0.90 MMP1 (0.78) MMP1MMP13MMP9MMP2MMP8
SCHEMBL6818064 0.90 MMP1 (0.78) MMP1MMP13MMP9MMP2MMP8
SCHEMBL6699509 0.89 MMP1 (0.84) MMP1MMP13MMP9MMP2MMP8
SCHEMBL6813091 0.88 MMP1 (0.76) MMP1MMP13MMP9MMP2MMP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 701 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1003720-B1 ARYLOXYARYLSULFONYLAMINO HYDROXAMIC ACID DERIVATIVES PFIZER PROD INC (US) 2004-03-31 EP claimed
US-6417229-B1 ENZYME INHIBITORS PFIZER INC 2002-07-09 US claimed
US-6214872-B1 ANTIARTHRITIC AND ANTICARCINOGENIC AGENTS PFIZER INC. 2001-04-10 US claimed
EP-1088550-A1 alpha-sulfonylamino hydroxamic acid inhibitors of matrix metallo-proteinases for the treatment of peripheral or central nervous system disorders Pfizer Products Inc. (US) 2001-04-04 EP claimed
EP-0930067-A2 MMP INHIBITORS FOR THE TREATMENT OF OCULAR ANGIOGENESIS Pfizer Products Inc. (US) 1999-07-21 EP claimed
JP-11263735-A None JP disclosed
US-20250320217-A1 SUBSTITUTED IMIDAZO[1,2-B]PYRIDAZINES AS PROTEIN KINASE INHIBITORS SUMITOMO PHARMA AMERICA INC (US) 2025-10-16 US disclosed
US-20250214963-A1 SULFONYL AMIDE DERIVATIVES FOR THE TREATMENT OF ABNORMAL CELL GROWTH PFIZER INC. 2025-07-03 US disclosed
US-20250129085-A1 SUBSTITUTED IMIDAZO[1,2-B]PYRIDAZINES AS PROTEIN KINASE INHIBITORS SUMITOMO PHARMA AMERICA INC (US) 2025-04-24 US disclosed
US-12037404-B2 Human monoclonal antibodies against EphA4 and their use THE HONG KONG UNIVERSITY OF SCIENCE AND TECHNOLOGY (CN) 2024-07-16 US disclosed
EP-2534153-B2 SALTS AND POLYMORPHS OF 8-FLUORO-2-{4-[(METHYLAMINO}METHYL]PHENYL}-1,3,4,5-TETRAHYDRO-6H-AZEPINO[5,4,3-CD]INDOL-6-ONE PFIZER (US) 2024-05-22 EP disclosed
US-20240109862-A1 SULFONYL AMIDE DERIVATIVES FOR THE TREATMENT OF ABNORMAL CELL GROWTH PFIZER INC. 2024-04-04 US disclosed
JP-2000026400-A PROCESS FOR ALKYLATION OF HINDERED SULFONAMIDE PFIZER PROD INC 2000-01-25 JP disclosed
WO-1999052862-A1 PROCESS FOR ALKYLATING HINDERED SULFONAMIDES USEFUL IN THE PRODUCTION OF MATRIX METALLOPROTEINASE INHIBITORS PFIZER PRODUCTS INC. (US) 1999-10-21 WO disclosed
EP-0949244-A2 Process for preparing hydroxamic acids Pfizer Products Inc. (US) 1999-10-13 EP disclosed
EP-0949245-A1 Process for alkylating hindered sulfonamides Pfizer Products Inc. (US) 1999-10-13 EP disclosed
EP-0949246-A1 Process for preparing phenoxyphenylsulfonyl halides Pfizer Products Inc. (US) 1999-10-13 EP disclosed
JP-H11263735-A USE OF MMP INHIBITOR FOR TREATMENT OF NEW EYEBALL VASCULOGENESIS PFIZER PROD INC 1999-09-28 JP disclosed
EP-0930067-A2 MMP INHIBITORS FOR THE TREATMENT OF OCULAR ANGIOGENESIS Pfizer Products Inc. (US) 1999-07-21 EP disclosed
WO-1999007675-A1 ARYLOXYARYLSULFONYLAMINO HYDROXAMIC ACID DERIVATIVES PFIZER PRODUCTS INC. (US) 1999-02-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250214963-A1 SULFONYL AMIDE DERIVATIVES FOR THE TREATMENT OF ABNORMAL CELL GROWTH GPR119, INSR, LYAR MMP1 3955/4885MMP13 4604/4885MMP9 4635/4885
US-20250129085-A1 SUBSTITUTED IMIDAZO[1,2-B]PYRIDAZINES AS PROTEIN KINASE INHIBITORS PIM1, PIM2, PIM3 MMP1 2061/4885MMP13 4280/4885MMP9 3879/4885
US-20240109862-A1 SULFONYL AMIDE DERIVATIVES FOR THE TREATMENT OF ABNORMAL CELL GROWTH GPR119, INSR, LYAR MMP1 3955/4885MMP13 4604/4885MMP9 4635/4885
US-20250320217-A1 SUBSTITUTED IMIDAZO[1,2-B]PYRIDAZINES AS PROTEIN KINASE INHIBITORS PIM1, PIM2, PIM3 MMP1 2061/4885MMP13 4280/4885MMP9 3879/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.