SCHEMBL6876876

SCHEMBL6876876

N#C[C@H](NC(=O)CCNC(=O)N1CCN(C(=O)O)CC1)SCc1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 6/20 0.43
MEN1 O00255 1/20 0.39
CNR1 P21554 1/20 0.39
CNR2 P34972 1/20 0.39
KMT2A Q03164 1/20 0.39
EPHX2 P34913 1/20 0.38
KDM4E B2RXH2 1/20 0.37
CHRM4 P08173 4/20 0.37
TPSAB1 Q15661 2/20 0.37
POLB P06746 2/20 0.36
ALDH1A1 P00352 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36
HRH3 Q9Y5N1 1/20 0.35
DPP4 P27487 1/20 0.35
DPP8 Q6V1X1 1/20 0.35
DPP7 Q9UHL4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5523224 0.88 ALDH1A1 (0.53) MEN1CNR1CNR2KMT2APOLB
SCHEMBL6876880 0.73 KDM4E (0.42) MEN1KMT2AKDM4EPOLBALDH1A1
SCHEMBL6876670 0.72 GAA (0.47) KMT2AALDH1A1CYP1A2CYP2C9
SCHEMBL6064318 0.69 NAMPT (0.39) NAMPTMEN1CNR1CNR2KMT2A
SCHEMBL18409626 0.69 PPARG (0.57)
SCHEMBL6742707 0.69 TSHR (0.50) MEN1KMT2APOLBALDH1A1CYP1A2
SCHEMBL5522704 0.68 GLS (0.44) NAMPTKMT2AALDH1A1
SCHEMBL6742151 0.68 STS (0.47) KDM4E
SCHEMBL6876870 0.67 CTSS (0.47) POLB
SCHEMBL5519770 0.67 PRMT5 (0.46) KMT2ACYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1452522-A2 Novel compounds and compositions as protease inhibitors AXYS PHARMACEUTICALS, INC. (US) 2004-09-01 EP disclosed