SCHEMBL6876880

SCHEMBL6876880

N#CCNC(=O)C(CNC(=O)N1CCN(C(=O)O)CC1)SCc1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.42
CTSS P25774 7/20 0.41
CTSK P43235 6/20 0.41
ALDH1A1 P00352 2/20 0.40
CYP1A2 P05177 1/20 0.40
POLB P06746 1/20 0.40
CYP2C9 P11712 1/20 0.40
CTSL P07711 6/20 0.40
CTSB P07858 4/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
SLC1A3 P43003 1/20 0.39
SLC1A2 P43004 1/20 0.39
PRMT5 O14744 1/20 0.37
WDR77 Q9BQA1 1/20 0.37
ATM Q13315 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5517777 0.89 CTSS (0.48) CTSSCTSKCTSLCTSB
SCHEMBL5523231 0.89 ALDH1A1 (0.56) KDM4EALDH1A1CYP1A2POLBCYP2C9
SCHEMBL5518404 0.87 POLB (0.52) KDM4EALDH1A1CYP1A2POLBCTSL
SCHEMBL5532239 0.87 CTSS (0.46) KDM4ECTSSCTSKALDH1A1CYP1A2
SCHEMBL6742393 0.82 CTSS (0.49) CTSSCTSKCTSLCTSBATM
SCHEMBL5524114 0.79 CTSL (0.56) CTSSCTSKCTSLCTSB
SCHEMBL6876870 0.78 CTSS (0.47) CTSSCTSKPOLBCTSLCTSB
SCHEMBL5520661 0.77 CTSS (0.46) CTSSCTSKCTSLCTSBMEN1
SCHEMBL5521867 0.77 ADRB1 (0.47) CTSSCTSKCYP2C9CTSLCTSB
SCHEMBL5527139 0.76 KDM4E (0.43) KDM4ECTSSALDH1A1POLBMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1452522-A2 Novel compounds and compositions as protease inhibitors AXYS PHARMACEUTICALS, INC. (US) 2004-09-01 EP disclosed