SCHEMBL687749

SCHEMBL687749

O=C(O)C[C@H](NC(=O)Nc1cccn(CCCOc2ccccc2)c1=O)c1ccc2c(c1)OCO2

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.48
ITGB3 P05106 9/20 0.42
ITGA2B P08514 7/20 0.42
CASP1 P29466 2/20 0.42
ITGAV P06756 3/20 0.41
NPC1 O15118 1/20 0.40
TP53 P04637 1/20 0.40
RAB9A P51151 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
EPHX2 P34913 1/20 0.40
KMT2A Q03164 2/20 0.39
MAOB P27338 1/20 0.39
MAPT P10636 1/20 0.38
ALOX15 P16050 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4757908 0.86 ITGB3 (0.42) GAAITGB3ITGA2BITGAVTP53
SCHEMBL687571 0.85 ALDH1A1 (0.50) ITGB3ITGA2BITGAVTP53SMN1; SMN2
SCHEMBL687727 0.83 POLB (0.44) ITGB3ITGA2BITGAVNPC1TP53
SCHEMBL687428 0.83 PTGER3 (0.56) ITGB3ITGAVRAB9ASMN1; SMN2KMT2A
SCHEMBL687886 0.83 PTGER3 (0.56) ITGB3ITGAVRAB9ASMN1; SMN2KMT2A
SCHEMBL688223 0.82 PTGER3 (0.55) GAACASP1TP53RAB9ASMN1; SMN2
SCHEMBL687922 0.82 PTGER3 (0.50) GAATP53KMT2A
SCHEMBL695420 0.82 MAPT (0.54) ITGB3ITGA2BTP53SMN1; SMN2KMT2A
SCHEMBL688325 0.82 ALDH1A1 (0.51) ITGB3ITGA2BITGAVTP53SMN1; SMN2
SCHEMBL687253 0.82 ITGB3 (0.44) ITGB3ITGA2BITGAV

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1203766-B1 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors ENCYSIVE PHARMACEUTICALS INC (US) 2012-02-29 EP disclosed