SCHEMBL6878265

SCHEMBL6878265

CN(C)c1nc(N[C@H]2CC[C@@H](NC(=O)Nc3cccs3)CC2)nc2c1CCCC2

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.53
HPGD P15428 2/20 0.53
GFER P55789 2/20 0.53
MAPT P10636 2/20 0.53
ALOX15 P16050 1/20 0.53
HSD17B10 Q99714 1/20 0.53
GAA P10253 2/20 0.53
RAB9A P51151 1/20 0.53
MCHR1 Q99705 16/20 0.40
ADRA2A P08913 13/20 0.40
HRH1 P35367 5/20 0.40
HTR2B P41595 5/20 0.40
ADRA1A P35348 3/20 0.40
HTR1A P08908 1/20 0.38
NPY5R Q15761 1/20 0.38
KDM4E B2RXH2 1/20 0.38
MEN1 O00255 1/20 0.38
LMNA P02545 1/20 0.38
HTT P42858 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6878270 1.00 ALDH1A1 (0.53) ALDH1A1HPGDGFERMAPTALOX15
SCHEMBL27652861 0.85 HPGD (0.50) ALDH1A1HPGDHSD17B10RAB9AMCHR1
SCHEMBL27652859 0.85 HPGD (0.50) ALDH1A1HPGDHSD17B10RAB9AMCHR1
SCHEMBL6878339 0.84 MCHR1 (0.41) HPGDMCHR1ADRA2AHRH1HTR2B
SCHEMBL6878333 0.84 MCHR1 (0.41) HPGDMCHR1ADRA2AHRH1HTR2B
SCHEMBL6879288 0.83 EPHX1 (0.53) MCHR1ADRA2AHRH1HTR2BADRA1A
SCHEMBL6879285 0.83 EPHX1 (0.53) MCHR1ADRA2AHRH1HTR2BADRA1A
SCHEMBL6872301 0.83 CYP3A4 (0.46) ALDH1A1MAPTHSD17B10RAB9AMCHR1
SCHEMBL6872308 0.83 CYP3A4 (0.46) ALDH1A1MAPTHSD17B10RAB9AMCHR1
SCHEMBL6878362 0.83 ADAM17 (0.40) RAB9AMCHR1ADRA2AHRH1HTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP disclosed