SCHEMBL6878472

SCHEMBL6878472

CN(C)c1nc(NC2CCC(NC(=S)Nc3cc([N+](=O)[O-])ccc3Cl)CC2)nc2c1CCCC2

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 3/20 0.44
MCHR1 Q99705 3/20 0.44
ALDH1A1 P00352 5/20 0.43
POLB P06746 1/20 0.43
RAB9A P51151 2/20 0.43
P2RX4 Q99571 1/20 0.42
P2RX7 Q99572 1/20 0.42
P2RX2 Q9UBL9 1/20 0.42
MAPT P10636 4/20 0.39
HPGD P15428 1/20 0.39
KMT2A Q03164 4/20 0.38
LMNA P02545 2/20 0.38
TDP1 Q9NUW8 1/20 0.38
MEN1 O00255 3/20 0.38
SMN1; SMN2 Q16637 1/20 0.37
NCOA3 Q9Y6Q9 1/20 0.37
NPY1R P25929 1/20 0.36
NPY2R P49146 1/20 0.36
PKM P14618 1/20 0.36
HRH1 P35367 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6878467 1.00 ADRA2A (0.44) ADRA2AMCHR1ALDH1A1POLBRAB9A
SCHEMBL6867652 0.94 ADRA2A (0.44) ADRA2AMCHR1ALDH1A1POLBMAPT
SCHEMBL6867647 0.94 ADRA2A (0.44) ADRA2AMCHR1ALDH1A1POLBMAPT
SCHEMBL6873057 0.90 ALDH1A1 (0.45) ADRA2AMCHR1ALDH1A1POLBRAB9A
SCHEMBL6873049 0.90 ALDH1A1 (0.45) ADRA2AMCHR1ALDH1A1POLBRAB9A
SCHEMBL6874051 0.89 L3MBTL1 (0.45) ADRA2AMCHR1ALDH1A1MAPTKMT2A
SCHEMBL6874045 0.89 L3MBTL1 (0.45) ADRA2AMCHR1ALDH1A1MAPTKMT2A
SCHEMBL6875749 0.88 MAPT (0.46) ADRA2AMCHR1ALDH1A1MAPTHPGD
SCHEMBL6875743 0.88 MAPT (0.46) ADRA2AMCHR1ALDH1A1MAPTHPGD
SCHEMBL7044478 0.87 MEN1 (0.43) ADRA2AMCHR1ALDH1A1POLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP disclosed