SCHEMBL6881271

SCHEMBL6881271

NC(=O)c1ccccc1Sc1ncc(C(F)(F)F)s1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT1 Q96EB6 1/20 0.47
MLYCD O95822 1/20 0.38
SCD O00767 2/20 0.36
PARP1 P09874 4/20 0.34
CDC7 O00311 1/20 0.34
ROCK2 O75116 1/20 0.34
MAP4K4 O95819 1/20 0.34
PIM1 P11309 1/20 0.34
PRKACA P17612 1/20 0.34
CDK7 P50613 1/20 0.34
CDK9 P50750 1/20 0.34
HIPK2 Q9H2X6 1/20 0.34
IRAK4 Q9NWZ3 1/20 0.34
MAPT P10636 2/20 0.33
CTNNB1 P35222 1/20 0.33
WNT3A P56704 1/20 0.33
LMNA P02545 1/20 0.33
HTT P42858 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC8 Q9BY41 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30810243 0.74 BCAT2 (0.42) SCDPARP1CDC7ROCK2MAP4K4
SCHEMBL6633089 0.72 SIRT1 (0.48) SIRT1SCDPARP1CDC7ROCK2
SCHEMBL3077375 0.71 SIRT1 (0.77) SIRT1PARP1IRAK4MAPTCTNNB1
SCHEMBL6630237 0.71 SIRT1 (0.53) SIRT1PARP1MAPTKMT2AALDH1A1
SCHEMBL6650786 0.68 SIRT1 (0.53) SIRT1MAPTKDM4EALDH1A1HPGD
SCHEMBL149060 0.67 SIRT1 (0.55) SIRT1PARP1IRAK4MAPTCTNNB1
SCHEMBL6633843 0.65 SIRT1 (0.53) SIRT1PARP1ROCK2MAP4K4PIM1
SCHEMBL1030659 0.65 SIRT1 (1.00) SIRT1MAPTCTNNB1LMNAKMT2A
SCHEMBL27839664 0.64 SIRT1 (0.60) SIRT1PARP1IRAK4MAPTCTNNB1
SCHEMBL6630850 0.64 SIRT1 (0.59) SIRT1MAPTKDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1381603-A2 QUINUCLIDINE-SUBSTITUEDARYL MOIETIES FOR TREATMENT OF DISEASE ( NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDS ) PHARMACIA & UPJOHN COMPANY (US) 2004-01-21 EP claimed
WO-2002016358-A2 QUINUCLIDINE-SUBSTITUTED ARYL MOIETIES FOR TREATMENT OF DISEASE (NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDS) PHARMACIA & UPJOHN COMPANY (US) 2002-02-28 WO claimed