SCHEMBL6882525

SCHEMBL6882525

O=C(Oc1ccccc1)N1CCCCC1

nearest known ligand 0.81

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.81
POLB P06746 1/20 0.81
KMT2A Q03164 6/20 0.81
SMN1; SMN2 Q16637 5/20 0.81
MEN1 O00255 4/20 0.81
LMNA P02545 1/20 0.81
NPSR1 Q6W5P4 1/20 0.81
NPC1 O15118 4/20 0.73
GAA P10253 2/20 0.65
RAB9A P51151 3/20 0.63
MAPT P10636 2/20 0.63
HTT P42858 2/20 0.63
MGLL Q99685 1/20 0.61
TSHR P16473 2/20 0.59
TP53 P04637 1/20 0.58
CYP3A4 P08684 1/20 0.58
MAPK1 P28482 1/20 0.58
ALOX15 P16050 1/20 0.58
ADORA2A P29274 1/20 0.57
ADORA1 P30542 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11480252 1.00 ALDH1A1 (0.81) ALDH1A1POLBKMT2ASMN1; SMN2MEN1
SCHEMBL1578826 0.98 ALDH1A1 (0.78) ALDH1A1POLBKMT2ASMN1; SMN2MEN1
SCHEMBL3077817 0.94 SMN1; SMN2 (0.72) ALDH1A1POLBKMT2ASMN1; SMN2MEN1
SCHEMBL5653225 0.93 ALDH1A1 (0.77) ALDH1A1POLBKMT2ASMN1; SMN2MEN1
SCHEMBL8845496 0.93 ALDH1A1 (0.77) ALDH1A1POLBKMT2ASMN1; SMN2MEN1
SCHEMBL8845129 0.91 KMT2A (0.73) ALDH1A1POLBKMT2ASMN1; SMN2MEN1
SCHEMBL11882343 0.90 MGLL (0.72) ALDH1A1POLBKMT2ASMN1; SMN2MEN1
SCHEMBL5650832 0.90 KMT2A (1.00) ALDH1A1POLBKMT2ASMN1; SMN2MEN1
SCHEMBL5646504 0.85 KMT2A (0.70) ALDH1A1POLBKMT2ASMN1; SMN2MEN1
SCHEMBL27780514 0.85 MGLL (0.66) ALDH1A1POLBKMT2ASMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 79 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108617386-B Ecological cultivation mode for leisure and sightseeing of persimmon orchard in mountainous region 湖北省农业科学院果树茶叶研究所 2020-06-16 CN claimed
CN-102918027-A Modulators of the gpr119 receptor and the treatment of disorders related thereto ARENA PHARM INC 2013-02-06 CN claimed
CN-1436175-A Cyclic lactams as inhibitors of A beta-protein production BRISTOL MYERS SQUIBB PHARMACEU (US) 2003-08-13 CN claimed
EP-0635004-B1 4-DIPHENYLMETHYL PIPERIDINE DERIVATIVES AND PROCESS FOR THEIR PREPARATION MERRELL PHARMA INC (US) 2002-07-17 EP claimed
WO-2024227104-A1 BIFUNCTIONAL COMPOUNDS FOR DEGRADING BRAF VIA UBIQUITIN PROTEOSOME PATHWAY NURIX THERAPEUTICS, INC. (US) 2024-10-31 WO disclosed
US-20240308976-A1 COMPOUNDS THAT MEDIATE PROTEIN DEGRADATION AND USES THEREOF MONTE ROSA THERAPEUTICS AG (CH) 2024-09-19 US disclosed
CN-116848238-A Macrocyclic complement factor B inhibitors 阿雷克森制药公司 2023-10-03 CN disclosed
CN-116589467-A Degradation of Bruton's Tyrosine Kinase (BTK) by conjugation of BTK inhibitors with E3 ligase ligands and methods of use thereof 百济神州有限公司 2023-08-15 CN disclosed
CN-116589466-A Degradation of Bruton's Tyrosine Kinase (BTK) by conjugation of BTK inhibitors with E3 ligase ligands and methods of use thereof 百济神州有限公司 2023-08-15 CN disclosed
WO-2023139199-A1 COMPOUNDS AND THEIR USE IN TREATING CANCER ASTRAZENECA AB (SE) 2023-07-27 WO disclosed
CN-116133658-A Novel compounds as inhibitors of histone deacetylase 6 and pharmaceutical compositions comprising the same 株式会社 钟根堂 2023-05-16 CN disclosed
WO-2023069708-A1 COMPOUNDS THAT MEDIATE PROTEIN DEGRADATION AND USES THEREOF MONTE ROSA THERAPEUTICS, INC. (US) 2023-04-27 WO disclosed
US-4408053-A ANALGESICS HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1983-10-04 US disclosed
US-4408054-A ANALGESTICS HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1983-10-04 US disclosed
EP-0080104-A2 3-(4-Piperidyl)-1,2-benzisoxazoles, process for the preparation thereof, and a pharmaceutical composition comprising the same HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1983-06-01 EP disclosed
EP-0079564-A1 3-(1-Substituted-4-piperidyl)-1,2-benzisoxazoles, a process for the preparation thereof, a pharmaceutical composition comprising the same, and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1983-05-25 EP disclosed
US-4355037-A ANALGESICS HOECHST-ROUSSEL PHARMACEUTICALS (US) 1982-10-19 US disclosed
US-4234484-A FROM ALKOXYLATED CYCLIC AMIDES USING AS A CATALYST A QUATERNARY AMMONIUM OR ALKALI METAL SALT OF TETRAFLUOROBORIC OR HEXAFLUOROPHOSPHORIC ACID HOECHST AKTIENGESELLSCHAFT (DE) 1980-11-18 US disclosed
US-4149941-A ELECTROLYTIC ALKOXYLATION HOECHST AKTIENGESELLSCHAFT (DE) 1979-04-17 US disclosed
US-4118500-A Fungicidal alkoxy mono- and dialkoxy N-substituted cyclic amines HOECHST AKTIENGESELLSCHAFT (DE) 1978-10-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240308976-A1 COMPOUNDS THAT MEDIATE PROTEIN DEGRADATION AND USES THEREOF CRBN, GSPT1, GSPT2 ALDH1A1 4088/4885POLB 4764/4885KMT2A 3669/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.