SCHEMBL6883723

SCHEMBL6883723

Cc1ccc(CN(C)C(=O)c2nc(-c3ccco3)[nH]c(=O)c2O)cc1Cl

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
RNASEH1 O60930 1/20 0.38
PIN1 Q13526 2/20 0.38
LMNA P02545 1/20 0.37
TP53 P04637 1/20 0.37
MAPT P10636 1/20 0.37
KDM4E B2RXH2 1/20 0.37
NPC1 O15118 1/20 0.37
ALDH1A1 P00352 1/20 0.37
HPGD P15428 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
POLB P06746 1/20 0.36
CDK4 P11802 1/20 0.36
CCND1 P24385 1/20 0.36
TMIGD3 P0DMS9 1/20 0.35
ADORA1 P30542 1/20 0.35
ERCC1 P07992 1/20 0.35
FEN1 P39748 1/20 0.35
ERCC4 Q92889 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6875960 0.93 RNASEH1 (0.44) RNASEH1PIN1LMNAMAPTKDM4E
SCHEMBL6884865 0.92 ALDH1A1 (0.39) PIN1LMNAMAPTKDM4ENPC1
SCHEMBL6877025 0.85 PIN1 (0.53) RNASEH1PIN1ERCC1FEN1ERCC4
SCHEMBL6884737 0.84 UBE2I (0.43) PIN1LMNAMAPTKDM4EALDH1A1
SCHEMBL6883616 0.83 PIN1 (0.40) RNASEH1PIN1ALDH1A1ERCC1FEN1
SCHEMBL6882673 0.82 ERCC1 (0.42) RNASEH1PIN1KDM4EALDH1A1HPGD
SCHEMBL6883326 0.82 ALDH1A1 (0.44) RNASEH1PIN1LMNAMAPTKDM4E
SCHEMBL6883865 0.82 PIN1 (0.40) RNASEH1PIN1ERCC1FEN1ERCC4
SCHEMBL6885416 0.81 HSP90AA1 (0.41) RNASEH1PIN1ERCC1FEN1ERCC4
SCHEMBL6883344 0.81 PIN1 (0.43) RNASEH1PIN1KDM4EALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004096128-A2 HIV INTEGRASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-11-11 WO claimed
WO-2004096128-A2 HIV INTEGRASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-11-11 WO disclosed