SCHEMBL6884865

SCHEMBL6884865

Cc1ccc(CN(C)C(=O)c2nc(-c3ccco3)[nH]c(=O)c2O)cc1C

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.39
HPGD P15428 3/20 0.39
POLB P06746 2/20 0.39
MAPT P10636 2/20 0.39
KDM4E B2RXH2 4/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
PIN1 Q13526 2/20 0.38
TMIGD3 P0DMS9 1/20 0.37
ADORA1 P30542 1/20 0.37
PKM P14618 1/20 0.37
ALOX15 P16050 1/20 0.37
TSHR P16473 1/20 0.37
ALOX12 P18054 1/20 0.37
HSD17B10 Q99714 1/20 0.37
ERCC1 P07992 1/20 0.36
FEN1 P39748 1/20 0.36
ERCC4 Q92889 1/20 0.36
OPRM1 P35372 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6883723 0.92 RNASEH1 (0.38) ALDH1A1HPGDPOLBMAPTKDM4E
SCHEMBL6875960 0.88 RNASEH1 (0.44) ALDH1A1MAPTKDM4ESMN1; SMN2PIN1
SCHEMBL6884737 0.86 UBE2I (0.43) ALDH1A1HPGDMAPTKDM4EPIN1
SCHEMBL6884889 0.84 PIN1 (0.55) PIN1ERCC1FEN1ERCC4
SCHEMBL6881498 0.82 PIN1 (0.39) PIN1ERCC1FEN1ERCC4
SCHEMBL6884690 0.81 PIN1 (0.44) ALDH1A1HPGDKDM4EPIN1TMIGD3
SCHEMBL6885506 0.81 ALDH1A1 (0.46) ALDH1A1HPGDMAPTKDM4ENPC1
SCHEMBL6885420 0.81 PIN1 (0.40) PIN1ERCC1FEN1ERCC4
SCHEMBL6883972 0.80 PIN1 (0.48) ALDH1A1HPGDKDM4ENPC1RAB9A
SCHEMBL6883275 0.80 RNASEH1 (0.40) PIN1ERCC1FEN1ERCC4MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004096128-A2 HIV INTEGRASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-11-11 WO claimed
WO-2004096128-A2 HIV INTEGRASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-11-11 WO disclosed