SCHEMBL6884629

SCHEMBL6884629

COc1ccc(-c2nc(C(=O)N(C)Cc3ccc(C)c(C)c3)c(O)c(=O)[nH]2)cc1

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ERCC1 P07992 2/20 0.44
FEN1 P39748 2/20 0.44
ERCC4 Q92889 2/20 0.44
TNKS O95271 1/20 0.43
PARP1 P09874 1/20 0.43
TNKS2 Q9H2K2 1/20 0.43
PIN1 Q13526 1/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
HSD17B2 P37059 2/20 0.41
HSP90AA1 P07900 2/20 0.40
HSP90AB1 P08238 1/20 0.40
CDKN1A P38936 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6883972 0.90 PIN1 (0.48) ERCC1FEN1ERCC4PIN1HSD17B2
SCHEMBL6884889 0.88 PIN1 (0.55) ERCC1FEN1ERCC4PIN1
SCHEMBL6886248 0.88 HSP90AA1 (0.46) ERCC1FEN1ERCC4PIN1MEN1
SCHEMBL6884690 0.87 PIN1 (0.44) ERCC1FEN1ERCC4PIN1
SCHEMBL6882799 0.87 ERCC1 (0.40) ERCC1FEN1ERCC4PIN1
SCHEMBL6883275 0.84 RNASEH1 (0.40) ERCC1FEN1ERCC4TNKSPIN1
SCHEMBL6886280 0.83 HTR7 (0.43) ERCC1FEN1ERCC4PIN1HSD17B2
SCHEMBL6883330 0.82 PIN1 (0.44) ERCC1FEN1ERCC4PIN1KMT2A
SCHEMBL6881498 0.80 PIN1 (0.39) ERCC1FEN1ERCC4PIN1
SCHEMBL6877025 0.80 PIN1 (0.53) ERCC1FEN1ERCC4PIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004096128-A2 HIV INTEGRASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-11-11 WO claimed
WO-2004096128-A2 HIV INTEGRASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-11-11 WO disclosed