SCHEMBL6884690

SCHEMBL6884690

Cc1ccc(CN(C)C(=O)c2nc(-c3ccncc3)[nH]c(=O)c2O)cc1C

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 2/20 0.44
ERCC1 P07992 3/20 0.44
FEN1 P39748 3/20 0.44
ERCC4 Q92889 3/20 0.44
HPGD P15428 2/20 0.42
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
HSD17B10 Q99714 1/20 0.42
RNASEH1 O60930 1/20 0.41
TMIGD3 P0DMS9 1/20 0.38
ADORA1 P30542 1/20 0.38
CHEK2 O96017 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6882673 0.91 ERCC1 (0.42) PIN1ERCC1FEN1ERCC4HPGD
SCHEMBL6884889 0.91 PIN1 (0.55) PIN1ERCC1FEN1ERCC4RNASEH1
SCHEMBL6883330 0.88 PIN1 (0.44) PIN1ERCC1FEN1ERCC4HPGD
SCHEMBL6884629 0.87 ERCC1 (0.44) PIN1ERCC1FEN1ERCC4
SCHEMBL6884051 0.87 RNASEH1 (0.46) PIN1ERCC1FEN1ERCC4HPGD
SCHEMBL6886274 0.85 ALOX5 (0.49) PIN1ERCC1FEN1ERCC4HPGD
SCHEMBL6885506 0.83 ALDH1A1 (0.46) PIN1HPGDKDM4EALDH1A1HSD17B10
SCHEMBL6883972 0.83 PIN1 (0.48) PIN1ERCC1FEN1ERCC4HPGD
SCHEMBL6882799 0.82 ERCC1 (0.40) PIN1ERCC1FEN1ERCC4RNASEH1
SCHEMBL6877025 0.82 PIN1 (0.53) PIN1ERCC1FEN1ERCC4RNASEH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004096128-A2 HIV INTEGRASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-11-11 WO claimed
WO-2004096128-A2 HIV INTEGRASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-11-11 WO disclosed