SCHEMBL688648

SCHEMBL688648

CN1C=C(C(=O)O)c2c(c3ccccc3n2C)C(C)(C)C1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.40
EGFR P00533 3/20 0.40
HSD17B10 Q99714 4/20 0.39
CYP2C19 P33261 1/20 0.39
ALDH1A1 P00352 8/20 0.39
MAPT P10636 3/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
NPC1 O15118 1/20 0.39
HTT P42858 1/20 0.39
RAB9A P51151 1/20 0.39
ATM Q13315 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
LMNA P02545 2/20 0.37
HK1 P19367 1/20 0.36
HKDC1 Q2TB90 1/20 0.36
SRC P12931 2/20 0.36
HPGD P15428 3/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL274281 0.83 ALDH1A1 (0.46) KDM4EHSD17B10ALDH1A1SMN1; SMN2NPC1
Bicarbonate SCHEMBL9678990 0.64 GPR3 (0.76) KDM4EEGFRHSD17B10ALDH1A1MAPT
SCHEMBL7487890 0.63 ALDH1A1 (0.70) KDM4EEGFRHSD17B10CYP2C19ALDH1A1
SCHEMBL7971242 0.63 MAPT (0.54) KDM4EEGFRHSD17B10CYP2C19ALDH1A1
SCHEMBL24010348 0.60 ALKBH5 (0.56) KDM4EEGFRHSD17B10ALDH1A1LMNA
SCHEMBL20595409 0.60 KDM4E (0.53) KDM4EEGFRHSD17B10ALDH1A1MAPT
SCHEMBL26031841 0.60 HSD17B10 (0.68) KDM4EEGFRHSD17B10CYP2C19ALDH1A1
SCHEMBL984736 0.59 EGFR (0.65) KDM4EEGFRHSD17B10CYP2C19ALDH1A1
SCHEMBL30443220 0.59 EGFR (0.65) KDM4EEGFRHSD17B10CYP2C19ALDH1A1
SCHEMBL5001736 0.59 ALDH1A1 (0.54) KDM4EEGFRHSD17B10CYP2C19ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1532153-B1 AZEPINOINDOLE AND PYRIDOINDOLE DERIVATIVES AS PHARMACEUTICAL AGENTS X CEPTOR THERAPEUTICS INC (US) 2012-02-29 EP disclosed