SCHEMBL6886679

SCHEMBL6886679

COc1ncc(Cl)cc1CN1CCC(C(C)c2ccccc2CCc2ccccc2)CC1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 1/20 0.38
MEN1 O00255 5/20 0.38
KMT2A Q03164 5/20 0.38
POLB P06746 1/20 0.37
DRD2 P14416 2/20 0.37
DRD4 P21917 2/20 0.37
HTR1A P08908 1/20 0.37
SLC6A4 P31645 1/20 0.37
ALDH1A1 P00352 1/20 0.36
ATM Q13315 1/20 0.36
SIGMAR1 Q99720 1/20 0.36
CXCR4 P61073 1/20 0.36
MAPT P10636 1/20 0.36
ALPL P05186 1/20 0.36
ALPI P09923 1/20 0.36
ALPG P10696 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5779587 0.86 DRD2 (0.42) MEN1KMT2APOLBDRD2DRD4
SCHEMBL6886685 0.82 DRD2 (0.47) DRD2DRD4
Oxalic Acid SCHEMBL5782031 0.76 MEN1 (0.41) MEN1KMT2APOLBALDH1A1MAPT
SCHEMBL5815276 0.75 KCNH2 (0.48) DRD2DRD4
SCHEMBL5780528 0.74 KCNH2 (0.45)
SCHEMBL5781339 0.74 MAOA (0.48) HTR1ASLC6A4ATM
SCHEMBL5778111 0.71 KCNH2 (0.50) DRD2DRD4
Oxalic Acid SCHEMBL5782849 0.70 KDM4E (0.41) MEN1KMT2AALDH1A1SIGMAR1MAPT
SCHEMBL5783805 0.70 MAOA (0.40) MCHR1MEN1KMT2AALDH1A1ATM
SCHEMBL5803181 0.70 DCPS (0.46) MEN1KMT2ADRD2DRD4ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6784192-B2 NA+ CHANNEL INHIBITORY ACTION IS USEFUL FOR THERAPY AND PREVENTION FOR EXAMPLE, ARRHYTHMIA, VARIOUS NEURALGIAS AND ANALGESIC EISAI CO., LTD. (JP) 2004-08-31 US disclosed
EP-1254904-A1 NOVEL PIPERIDINE COMPOUNDS AND DRUGS CONTAINING THE SAME Eisai Co., Ltd. (JP) 2002-11-06 EP disclosed