SCHEMBL6888239

SCHEMBL6888239

NC(=S)c1ccc(Br)cc1C(F)(F)F

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 2/20 0.44
DGAT1 O75907 1/20 0.42
ALDH1A1 P00352 2/20 0.41
NPFFR1 Q9GZQ6 1/20 0.39
NPFFR2 Q9Y5X5 1/20 0.39
CES2 O00748 1/20 0.38
PTPN7 P35236 1/20 0.35
DUSP3 P51452 1/20 0.35
CTSL P07711 3/20 0.35
EPRS1 P07814 1/20 0.34
CTSB P07858 1/20 0.34
HRH4 Q9H3N8 1/20 0.33
HPGD P15428 1/20 0.33
RAD52 P43351 1/20 0.33
HCAR1 Q9BXC0 1/20 0.32
TMPRSS4 Q9NRS4 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CA5A P35218 1/20 0.32
CA9 Q16790 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31231675 0.85 ALDH1A1 (0.44) KDM1ADGAT1ALDH1A1NPFFR1NPFFR2
SCHEMBL1330833 0.81 DGAT1 (0.59) KDM1ADGAT1NPFFR1NPFFR2CES2
SCHEMBL16527182 0.79 IDO1 (0.43) ALDH1A1CES2HPGDRAD52
SCHEMBL29333933 0.78 CES2 (0.46) KDM1ADGAT1CES2EPRS1HPGD
SCHEMBL6893498 0.78 GAA (0.41) ALDH1A1CES2TMPRSS4
SCHEMBL257339 0.77 EPRS1 (0.51) KDM1ADGAT1ALDH1A1CES2EPRS1
SCHEMBL28299420 0.77 KDM1A (0.42) KDM1ADGAT1NPFFR1NPFFR2CES2
SCHEMBL29451092 0.77 EPRS1 (0.51) KDM1ADGAT1ALDH1A1CES2EPRS1
SCHEMBL8479105 0.76 KDM1A (0.35) KDM1ADGAT1ALDH1A1NPFFR1NPFFR2
SCHEMBL25532291 0.76 CES2 (0.47) KDM1ADGAT1CES2EPRS1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1126833-A4 OXADIAZOLE, THIADIAZOLE AND TRIAZOLE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF TREGA BIOSCIENCES INC (US) 2004-09-08 EP claimed
EP-1126833-A2 OXADIAZOLE, THIADIAZOLE AND TRIAZOLE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF TREGA BIOSCIENCES, INC. (US) 2001-08-29 EP claimed
WO-2000025768-A1 OXADIAZOLE, THIADIAZOLE AND TRIAZOLE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF TREGA BIOSCIENCES, INC. (US) 2000-05-11 WO claimed