SCHEMBL6889135

SCHEMBL6889135

COC(=O)c1ccc(-c2cccc(O)c2)cc1C

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 8/20 0.54
HSD17B2 P37059 8/20 0.54
CA12 O43570 2/20 0.51
CA1 P00915 2/20 0.51
CA2 P00918 2/20 0.51
CA7 P43166 2/20 0.51
CA9 Q16790 2/20 0.51
CA14 Q9ULX7 2/20 0.51
PDK2 Q15119 1/20 0.51
PDK4 Q16654 1/20 0.51
CYP3A4 P08684 3/20 0.48
CYP2C9 P11712 1/20 0.48
EGFR P00533 2/20 0.46
SLC2A1 P11166 1/20 0.45
CYP2D6 P10635 2/20 0.44
CYP2C19 P33261 2/20 0.44
HPGDS O60760 1/20 0.43
ERN1 O75460 1/20 0.43
NR4A2 P43354 1/20 0.43
MEN1 O00255 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2884545 0.87 KDM4E (0.52) CA12CA1CA2CA7CA9
SCHEMBL28675075 0.85 CA12 (0.56) HSD17B1CA12CA1CA2CA7
SCHEMBL14084580 0.85 EGFR (0.56) EGFRSLC2A1NR4A2MEN1ALDH1A1
SCHEMBL25603748 0.83 SLC6A3 (0.47) CA12CA1CA2CA9EGFR
SCHEMBL3200407 0.83 GAA (0.51) CA12CA1CA2CA9EGFR
SCHEMBL31337006 0.82 EGFR (0.65) HSD17B1HSD17B2CA12CA1CA2
SCHEMBL6564981 0.82 HSD17B1 (0.59) HSD17B1HSD17B2CYP3A4CYP2C9EGFR
SCHEMBL4700092 0.82 EGFR (0.65) HSD17B1HSD17B2CA12CA1CA2
SCHEMBL131661 0.81 CA12 (0.69) CA12CA1CA2CA7CA9
SCHEMBL9150203 0.80 RXRB (0.57) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6831106-B1 Selective activity on cell proliferation and differentiation without displaying any hypercalcaemiant nature GALDERMA RESEARCH & DEVELOPMENT, S.N.C. (FR) 2004-12-14 US disclosed