SCHEMBL6890765

SCHEMBL6890765

NC(=S)c1ccc(OCc2ccccc2)cc1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP10 Q53GL7 2/20 0.70
NR4A1 P22736 1/20 0.64
NR4A2 P43354 1/20 0.64
NR4A3 Q92570 1/20 0.64
CYP1A2 P05177 2/20 0.61
CYP2C19 P33261 2/20 0.61
LMNA P02545 1/20 0.61
PTGS1 P23219 1/20 0.61
SLC6A2 P23975 1/20 0.61
PTGS2 P35354 1/20 0.61
SLC6A3 Q01959 1/20 0.61
HIF1A Q16665 1/20 0.61
HDAC6 Q9UBN7 1/20 0.61
RAB9A P51151 2/20 0.60
NPC1 O15118 1/20 0.60
CASP3 P42574 1/20 0.60
SENP8 Q96LD8 1/20 0.60
SENP7 Q9BQF6 1/20 0.60
SENP6 Q9GZR1 1/20 0.60
MAOB P27338 3/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7897887 0.83 NPC1 (0.62) PARP10RAB9ANPC1MAOBMAOA
SCHEMBL11119945 0.83 NR4A2 (0.64) PARP10NR4A2LMNARAB9ANPC1
SCHEMBL8558672 0.83 NPC1 (0.64) PARP10RAB9ANPC1MAOBMAPT
SCHEMBL27604519 0.82 MAOB (0.70) PARP10NR4A1NR4A2NR4A3CYP1A2
SCHEMBL119689 0.82 PARP10 (1.00) PARP10NR4A1NR4A2NR4A3CYP1A2
SCHEMBL6629683 0.82 F2 (0.83) PARP10F2PRSS1PRSS2PRSS3
SCHEMBL864192 0.81 ALDH1A1 (0.60) PARP10NR4A1NR4A2NR4A3CYP1A2
SCHEMBL6893845 0.81 NR4A2 (0.67) NR4A2MAOBSRD5A2F2
SCHEMBL28017864 0.81 FFAR1 (0.56) PARP10LMNARAB9ANPC1PLA2G4B
SCHEMBL521489 0.81 NR4A1 (0.72) PARP10NR4A1NR4A2NR4A3CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1126833-A4 OXADIAZOLE, THIADIAZOLE AND TRIAZOLE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF TREGA BIOSCIENCES INC (US) 2004-09-08 EP claimed
EP-1126833-A2 OXADIAZOLE, THIADIAZOLE AND TRIAZOLE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF TREGA BIOSCIENCES, INC. (US) 2001-08-29 EP claimed
WO-2000025768-A1 OXADIAZOLE, THIADIAZOLE AND TRIAZOLE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF TREGA BIOSCIENCES, INC. (US) 2000-05-11 WO claimed
CN-104817553-B The pyrimidinediamine class compound and its derivative and its medical usage of a kind of aromatic radical-heterocyclic substituted 华东师范大学 2018-11-09 CN disclosed
CN-103694195-B Aromatic heterocyclic small molecular organic compounds and derivative, preparation method and medicinal use EAST CHINA NORMAL UNIVERSITY (CN) 2016-04-06 CN disclosed
CN-104817553-A Aryl-heterocycle substituted pyrimidinediamine compound and its derivative and pharmaceutical use thereof UNIV EAST CHINA NORMAL 2015-08-05 CN disclosed
CN-103694195-A Heterocyclic aromatic micromolecule organic compounds and derivatives, preparation method and medical application UNIV EAST CHINA NORMAL 2014-04-02 CN disclosed
US-6191289-B1 REACTING A 4-OXO-4H-BENZOPYRAN GROUP SUBSTITUTED WITH AMIDE OR A PHENYL GROUP IN ITS 2 POSITION IS REACTED WITH ANHYDROUS HYDRAZINE OR SALT IN PRESENCE OF CATALYST FOLLOWED BY REACTING WITH NITROUS ACID OR SALT TO FORM TETRAZOLE COMPOUND SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2001-02-20 US disclosed
US-5874593-A SULFUR CONTAINING AMIDE SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1999-02-23 US disclosed
EP-0711762-A1 PROCESS FOR PRODUCING TETRAZOLE COMPOUND AND INTERMEDIATE THEREFOR SUMITOMO CHEMICAL COMPANY LIMITED (JP) 1996-05-15 EP disclosed