SCHEMBL6892450

SCHEMBL6892450

Cc1ccc(Cc2cc(C(=O)NC3CCCCC3)nc3ccccc23)cn1

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 2/20 0.54
RAB9A P51151 1/20 0.53
ADAM17 P78536 1/20 0.49
TP53 P04637 1/20 0.48
GAA P10253 1/20 0.47
KMT2A Q03164 1/20 0.47
RXFP1 Q9HBX9 4/20 0.47
LMNA P02545 2/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
KDM4E B2RXH2 1/20 0.46
ALDH1A1 P00352 1/20 0.46
ALOX5 P09917 1/20 0.46
CYP2C9 P11712 1/20 0.46
KCNH2 Q12809 1/20 0.46
MAPT P10636 2/20 0.46
MAPK1 P28482 2/20 0.46
USP2 O75604 1/20 0.46
RECQL P46063 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2224496 0.88 GAA (0.55) CHRM1RAB9AGAAKMT2ARXFP1
SCHEMBL6890076 0.88 KCNH2 (0.48) RAB9ATP53GAAKMT2ARXFP1
SCHEMBL2275863 0.88 CHRM1 (0.70) CHRM1ADAM17ALOX5CYP2C9KCNH2
SCHEMBL6891717 0.87 CHRM1 (0.54) CHRM1RAB9AADAM17TP53GAA
SCHEMBL6893880 0.87 CHRM1 (0.54) CHRM1RAB9AGAAKMT2ARXFP1
SCHEMBL6891135 0.87 CHRM1 (0.57) CHRM1RAB9AADAM17ALOX5CYP2C9
SCHEMBL6891970 0.86 GAA (0.49) RAB9ATP53GAAKMT2ARXFP1
SCHEMBL18756570 0.86 CHRM1 (0.46) CHRM1RAB9AKMT2ALMNASMN1; SMN2
SCHEMBL6890115 0.86 GAA (0.45) RAB9ATP53GAAKMT2ARXFP1
SCHEMBL17656777 0.85 CHRM1 (0.51) CHRM1RAB9ALMNASMN1; SMN2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011084368-A1 QUINOLINE AMIDE M1 RECEPTOR POSITIVE ALLOSTERIC MODULATORS MERCK SHARP & DOHME CORP. (US) 2011-07-14 WO disclosed