SCHEMBL6894752

SCHEMBL6894752

O=S(=O)(Cl)c1cc(F)c(Br)c(Br)c1F

nearest known ligand 0.32

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TRPV4 Q9HBA0 1/20 0.32
CA12 O43570 1/20 0.30
CA1 P00915 1/20 0.30
CA2 P00918 1/20 0.30
CA7 P43166 1/20 0.30
CA13 Q8N1Q1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6675574 0.79 CA12 (0.34) TRPV4CA12CA1CA2CA7
SCHEMBL29671274 0.76 CA12 (0.38) TRPV4CA12CA1CA2CA7
SCHEMBL1535900 0.76 CA12 (0.38) TRPV4CA12CA1CA2CA7
SCHEMBL28006505 0.75 CES2 (0.33) TRPV4
SCHEMBL4206943 0.75 TRPV4 (0.35) TRPV4
SCHEMBL6674733 0.72 TRPV4 (0.32) TRPV4CA12CA1CA2CA7
SCHEMBL384682 0.72 PKM (0.38) TRPV4CA12CA1CA2CA7
SCHEMBL29835220 0.72 PKM (0.38) TRPV4CA12CA1CA2CA7
SCHEMBL1541882 0.71 CA1 (0.41) CA12CA1CA2CA7
SCHEMBL699765 0.71 CA12 (0.34) TRPV4CA12CA1CA2CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1126833-A4 OXADIAZOLE, THIADIAZOLE AND TRIAZOLE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF TREGA BIOSCIENCES INC (US) 2004-09-08 EP disclosed
EP-1126833-A2 OXADIAZOLE, THIADIAZOLE AND TRIAZOLE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF TREGA BIOSCIENCES, INC. (US) 2001-08-29 EP disclosed
WO-2000025768-A1 OXADIAZOLE, THIADIAZOLE AND TRIAZOLE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF TREGA BIOSCIENCES, INC. (US) 2000-05-11 WO disclosed