SCHEMBL6895816

SCHEMBL6895816

C[C@@H](O)[C@@H](N)C(NCc1cccc(C(F)(F)F)c1)c1cc(F)cc(F)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.48
HTR2B P41595 2/20 0.48
HTR2C P28335 1/20 0.48
SIGMAR1 Q99720 2/20 0.43
LMNA P02545 1/20 0.43
MAPT P10636 1/20 0.43
ADRA2C P18825 1/20 0.43
SLC6A4 P31645 1/20 0.43
ADRA1A P35348 1/20 0.43
DRD3 P35462 1/20 0.43
OPRK1 P41145 1/20 0.43
EPHX1 P07099 2/20 0.40
IDO1 P14902 2/20 0.40
BCHE P06276 2/20 0.39
TP53 P04637 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
TSHR P16473 1/20 0.39
CYP2C19 P33261 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL164926 0.88 HTR2A (0.50) HTR2AHTR2BHTR2CSIGMAR1LMNA
SCHEMBL5578711 0.87 BACE1 (0.35)
SCHEMBL6887215 0.87 MAOB (0.41) IDO1
SCHEMBL6895217 0.84 SIGMAR1 (0.40) SIGMAR1LMNAIDO1CYP1A2CYP2D6
SCHEMBL6889713 0.84 MEN1 (0.40) SIGMAR1IDO1CYP1A2CYP2D6CYP2C19
SCHEMBL6894740 0.82 TAAR1 (0.46) LMNAIDO1CASR
SCHEMBL6895046 0.81 IDO1 (0.33) IDO1
SCHEMBL6894401 0.81 MEN1 (0.39)
SCHEMBL6887059 0.79 TACR1 (0.50)
SCHEMBL3645149 0.78 BCHE (0.52) HTR2AHTR2BHTR2CBCHECASR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2004502669-A 2004-01-29 JP claimed
EP-1353898-A2 COMPOUNDS TO TREAT ALZHEIMER'S DISEASE Elan Pharmaceuticals, Inc. (US) 2003-10-22 EP claimed
WO-2002002512-A2 COMPOUNDS TO TREAT ALZHEIMER'S DISEASE ELAN PHARMACEUTICALS, INC. (US) 2002-01-10 WO claimed