SCHEMBL6897129

SCHEMBL6897129

COc1cc(CC(=O)O)cc(OC)c1OC.O=C(O)CCC(=O)c1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NR4A2 P43354 1/20 0.54
ALDH1A1 P00352 5/20 0.50
GAA P10253 3/20 0.50
CYP2C19 P33261 2/20 0.50
TSHR P16473 1/20 0.48
NFKB1 P19838 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
CYP1A2 P05177 3/20 0.46
TP53 P04637 1/20 0.46
SMN1; SMN2 Q16637 3/20 0.45
KDM4E B2RXH2 2/20 0.45
LMNA P02545 2/20 0.45
FFAR1 O14842 1/20 0.45
RAB9A P51151 1/20 0.45
HIF1A Q16665 1/20 0.45
HPGD P15428 1/20 0.45
HSD17B10 Q99714 1/20 0.45
ATM Q13315 1/20 0.44
PTGDR2 Q9Y5Y4 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1983304 0.86 LMNA (0.54) ALDH1A1CYP1A2TP53SMN1; SMN2KDM4E
SCHEMBL6897135 0.84 LMNA (0.45) ALDH1A1TDP1CYP1A2TP53SMN1; SMN2
SCHEMBL499116 0.82 GAA (0.61) ALDH1A1GAATSHRNFKB1TDP1
SCHEMBL6822746 0.81 MAPK1 (0.56) ALDH1A1GAACYP2C19CYP1A2SMN1; SMN2
Hydrochloric Acid SCHEMBL4002124 0.81 GAA (0.59) ALDH1A1GAATSHRNFKB1TDP1
SCHEMBL27961458 0.77 ALDH1A1 (0.50) ALDH1A1CYP1A2TP53SMN1; SMN2KDM4E
SCHEMBL29141728 0.74 PTPN1 (0.52) ALDH1A1GAATSHRNFKB1TDP1
SCHEMBL9828028 0.74 MEN1 (0.62) ALDH1A1GAASMN1; SMN2KDM4E
SCHEMBL7823257 0.74 ALDH1A1 (0.61) ALDH1A1TDP1CYP1A2SMN1; SMN2KDM4E
SCHEMBL6926630 0.74 MEN1 (0.64) ALDH1A1GAATP53SMN1; SMN2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1126833-A4 OXADIAZOLE, THIADIAZOLE AND TRIAZOLE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF TREGA BIOSCIENCES INC (US) 2004-09-08 EP disclosed
EP-1126833-A2 OXADIAZOLE, THIADIAZOLE AND TRIAZOLE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF TREGA BIOSCIENCES, INC. (US) 2001-08-29 EP disclosed
WO-2000025768-A1 OXADIAZOLE, THIADIAZOLE AND TRIAZOLE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF TREGA BIOSCIENCES, INC. (US) 2000-05-11 WO disclosed