SCHEMBL6901679

SCHEMBL6901679

COC(=O)/C(=C/C(=O)O)C(=O)O

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 1/20 0.37
KDM4E B2RXH2 2/20 0.36
TSHR P16473 1/20 0.36
ALDH1A1 P00352 2/20 0.35
HTT P42858 1/20 0.34
MAPT P10636 3/20 0.33
EGLN1 Q9GZT9 1/20 0.33
LMNA P02545 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
HPGD P15428 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3277564 0.83 HCAR2 (0.36) HCAR2KDM4EALDH1A1MAPTEGLN1
SCHEMBL4596276 0.83 HCAR2 (0.42) HCAR2KDM4EALDH1A1MAPTEGLN1
SCHEMBL17235833 0.79 ALDH1A1 (0.38) HCAR2ALDH1A1MAPTEGLN1HPGD
SCHEMBL17287328 0.79 ALDH1A1 (0.38) HCAR2ALDH1A1MAPTEGLN1HPGD
SCHEMBL17138384 0.74 TSHR (0.41) KDM4ETSHRALDH1A1HTTMAPT
SCHEMBL269971 0.74 TSHR (0.41) KDM4ETSHRALDH1A1HTTMAPT
SCHEMBL599552 0.72 ALDH1A1 (0.42) HCAR2KDM4ETSHRALDH1A1HTT
SCHEMBL7771328 0.72 ALDH1A1 (0.42) HCAR2KDM4ETSHRALDH1A1HTT
SCHEMBL599554 0.72 ALDH1A1 (0.42) HCAR2KDM4ETSHRALDH1A1HTT
SCHEMBL8846164 0.72 TSHR (0.39) KDM4ETSHRALDH1A1HTTMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0734401-B1 APPARATUS AND PROCESS FOR THE PRODUCTION OF LOW MOLECULAR WEIGHT GRAFTED POLYOLEFINS EASTMAN CHEM CO (US) 1997-10-29 EP claimed
EP-0734401-A1 APPARATUS AND PROCESS FOR THE PRODUCTION OF LOW MOLECULAR WEIGHT GRAFTED POLYOLEFINS EASTMAN CHEM CO (US) 1996-10-02 EP claimed
WO-1995016717-A1 APPARATUS AND PROCESS FOR THE PRODUCTION OF LOW MOLECULAR WEIGHT GRAFTED POLYOLEFINS EASTMAN CHEMICAL COMPANY (US) 1995-06-22 WO claimed
WO-1995016719-A1 LOW MOLECULAR WEIGHT GRAFTED RANDOM ETHYLENE/PROPYLENE COPOLYMER OF HIGH ACID NUMBER AND METHOD FOR PREPARATION THEREOF EASTMAN CHEMICAL COMPANY (US) 1995-06-22 WO claimed
EP-1230300-B1 OLEFINIC SLIP-COATING FOR AUTOMOTIVE WEATHERSEALS ADVANCED ELASTOMER SYSTEMS (US) 2004-07-14 EP disclosed
US-6602589-B2 Formed by extrusion of an olefin-based thermoplastic elastomer or vulcanizate; contains a novel compatibilizer which allows thermoplastic polyurethane to bond to graft polymer of polypropylene ADVANCED ELASTOMER SYSTEMS, L.P. 2003-08-05 US disclosed
US-20020091182-A1 Olefinic slip-coating for automotive weatherseals EXXONMOBIL CHEMICAL PATENTS INC. 2002-07-11 US disclosed
US-6368700-B1 BLEND OF UNSATURATED POLYER, THERMOPLASTIC POLYURETHANE AND ALPHA-OLEFIN ADVANCED ELASTOMER SYSTEMS, L.P. 2002-04-09 US disclosed
US-6187870-B1 Apparatus and process for the production of low molecular weight grafted polyolefins EASTMAN CHEMICAL COMPANY 2001-02-13 US disclosed
US-6166118-A Emulsification process for functionalized polyolefins and emulsions made therefrom EASTMAN CHEMICAL COMPANY (US) 2000-12-26 US disclosed
EP-0734401-B1 APPARATUS AND PROCESS FOR THE PRODUCTION OF LOW MOLECULAR WEIGHT GRAFTED POLYOLEFINS EASTMAN CHEM CO (US) 1997-10-29 EP disclosed
WO-1995021204-A1 CHLOROSULFONATED ETHYLENE ALPHA-OLEFIN GRAFT POLYMERS E.I. DU PONT DE NEMOURS AND COMPANY (US) 1995-08-10 WO disclosed
WO-1995016719-A1 LOW MOLECULAR WEIGHT GRAFTED RANDOM ETHYLENE/PROPYLENE COPOLYMER OF HIGH ACID NUMBER AND METHOD FOR PREPARATION THEREOF EASTMAN CHEMICAL COMPANY (US) 1995-06-22 WO disclosed
EP-0633301-A2 Modified halogenated polyolefin adhesives LORD CORPORATION (US) 1995-01-11 EP disclosed
EP-0489495-A2 Modified halogenated polyolefin adhesives LORD CORPORATION (US) 1992-06-10 EP disclosed
US-5102956-A Graft with acid anhydride, modified by polyhydroxylic aromatic compound and sulfur containing compounds to improved peel strength LORD CORPORATION (US) 1992-04-07 US disclosed
US-4822688-A PROPYLENE-ANHYDRIDE GRAFT POLYMER REACTED WITH DIAMINE NOGUES PIERRE (FR) 1989-04-18 US disclosed
US-4735992-A COATINGS FOR METALS SOCIETE ATOCHEM (FR) 1988-04-05 US disclosed
US-4727120-A MALEIC ANHYDRIDE AND DIOL GRAFT POLYMERS SOCIETE ATOCHEM (FR) 1988-02-23 US disclosed