SCHEMBL6903725

SCHEMBL6903725

CCOC(=O)C(c1ccccc1)(c1ccccc1)N1CCCCC1

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP2B6 P20813 1/20 0.46
PIN1 Q13526 1/20 0.44
ALDH1A1 P00352 4/20 0.44
MAPT P10636 2/20 0.44
CHRM3 P20309 7/20 0.43
NPSR1 Q6W5P4 1/20 0.43
CCR1 P32246 1/20 0.41
CHRM2 P08172 1/20 0.40
CHRM4 P08173 1/20 0.40
CHRM5 P08912 1/20 0.40
CYP2D6 P10635 1/20 0.40
CHRM1 P11229 1/20 0.40
RECQL P46063 1/20 0.40
TSHR P16473 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7559824 0.83 KCNN4 (0.51) CYP2B6ALDH1A1MAPTCHRM3NPSR1
SCHEMBL10982647 0.78 CHRM3 (0.46) PIN1ALDH1A1MAPTCHRM3CHRM2
SCHEMBL7646732 0.74 PIN1 (0.54) PIN1ALDH1A1MAPTCHRM3NPSR1
SCHEMBL4525774 0.73 CYP2B6 (0.47) CYP2B6MAPTCHRM3CHRM2CYP2D6
SCHEMBL1647761 0.72 KCNN4 (0.62) PIN1ALDH1A1MAPTCHRM3NPSR1
SCHEMBL5639395 0.72 PIN1 (0.56) PIN1ALDH1A1MAPTCHRM3NPSR1
SCHEMBL26039065 0.72 ALDH1A1 (0.39) ALDH1A1MAPTCYP2D6TSHR
SCHEMBL27916287 0.71 CES1 (0.56) PIN1ALDH1A1MAPTCHRM3NPSR1
SCHEMBL2128439 0.71 CYP2B6 (0.50) CYP2B6CHRM3NPSR1CHRM2CHRM4
SCHEMBL2127685 0.71 CYP2B6 (0.50) CYP2B6CHRM3NPSR1CHRM2CHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6797694-B2 TRIARYLMETHANE DERIVATIVES HAVING INHIBITORY ACTIVITY ON AN INTERMEDIATE CONDUCTANCE CALCIUM ION ACTIVATED POTASSIUM CHANNEL (IKCA) POSEIDON PHARMACEUTICALS A/S (DK) 2004-09-28 US claimed
US-20020065247-A1 Chemical compounds having ion channel blocking activity for the treatment of immune dysfunction NEUROSEARCH A/S (DK) 2002-05-30 US claimed
EP-1181016-A1 CHEMICAL COMPOUNDS HAVING ION CHANNEL BLOCKING ACTIVITY FOR THE TREATMENT OFIMMUNE DYSFUNCTION NEUROSEARCH A/S (DK) 2002-02-27 EP claimed
WO-2000069439-A1 CHEMICAL COMPOUNDS HAVING ION CHANNEL BLOCKING ACTIVITY FOR THE TREATMENT OF IMMUNE DYSFUNCTION NEUROSEARCH A/S (DK) 2000-11-23 WO claimed
US-7531573-B2 potent, selective and safe inhibitors of the Ca2+-activated potassium channel CHILDREN'S MEDICAL CENTER CORPORATION (US) 2009-05-12 US disclosed
US-7531573-B2 potent, selective and safe inhibitors of the Ca2+-activated potassium channel CHILDREN'S MEDICAL CENTER CORPORATION (US) 2009-05-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020065247-A1 Chemical compounds having ion channel blocking activity for the treatment of immune dysfunction KCNN2, KCNN1, KCNN3 CYP2B6 3761/4885PIN1 2990/4885ALDH1A1 2384/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.