SCHEMBL6906137

SCHEMBL6906137

Cc1ccc(S(=O)(=O)O)c(C[C@@H]2COc3ccc4nocc4c3O2)c1.O=C(c1ccc(F)cc1)C1CCN(CC2COc3ccc4nocc4c3O2)CC1

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 4/20 0.39
HTR2A P28223 4/20 0.38
HTR2C P28335 2/20 0.38
DRD2 P14416 1/20 0.38
HTR2B P41595 1/20 0.38
ALDH1A1 P00352 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
LMNA P02545 2/20 0.34
HSD11B1 P28845 2/20 0.34
HRH1 P35367 1/20 0.34
GAA P10253 1/20 0.34
HTT P42858 1/20 0.34
POLB P06746 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6797367 0.86 HTR2A (0.43) HTR1AHTR2AHTR2CDRD2HTR2B
SCHEMBL6906280 0.76 HTR1A (0.61) HTR1AHTR2AHTR2CDRD2HTR2B
SCHEMBL7247392 0.73 HTR1A (0.42) HTR1A
SCHEMBL6782174 0.73 HTR2A (0.51) HTR1AHTR2AHTR2CDRD2HTR2B
SCHEMBL6630732 0.71 HTR1A (0.46) HTR1ADRD2LMNAGAA
SCHEMBL6109572 0.71 HTR1A (0.46) HTR1ADRD2LMNAGAA
SCHEMBL4335129 0.71 NR3C1 (0.37) HTR1AALDH1A1SMN1; SMN2LMNAGAA
SCHEMBL7236260 0.70 CA2 (0.35) HTR1A
SCHEMBL7240006 0.70 CA2 (0.35) HTR1A
SCHEMBL6630585 0.70 HTR1A (0.39) HTR1ADRD2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6800642-B2 SUCH AS BENZYL-(-7,8-DIHYDRO-2,6,9-TRIOXA-3-AZA-CYCLOPENTA(A)NAPHTHALEN-8-YLMETHYL) -AMINE; FOR TREATMENT OF DRUG DEPENDENCE/ADDICTION, BIPOLAR DISORDER, PARKINSON'S DISEASE, LEVODOPA INDUCED PSYCHOSES OR DYSKINESIAS WYETH 2004-10-05 US disclosed