SCHEMBL6907017

SCHEMBL6907017

C=C(C)c1cc(CN(C)Cc2ccc(C(C)(C)C)cc2)cc(C(=C)C)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.46
SIGMAR1 Q99720 2/20 0.46
KCNH2 Q12809 2/20 0.46
CYP2D6 P10635 2/20 0.46
NR1I2 O75469 1/20 0.46
ADRA2A P08913 1/20 0.46
ACHE P22303 1/20 0.46
SLC6A2 P23975 1/20 0.46
HTR2A P28223 1/20 0.46
SLC6A4 P31645 1/20 0.46
TMEM97 Q5BJF2 1/20 0.40
NR1H4 Q96RI1 4/20 0.37
EPHX2 P34913 2/20 0.37
ESRRG P62508 1/20 0.36
HDAC3 O15379 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
TP53 P04637 1/20 0.35
CYP1A2 P05177 2/20 0.35
CYP2C19 P33261 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6910551 0.92 LMNA (0.42) LMNASIGMAR1KCNH2CYP2D6NR1I2
SCHEMBL6914310 0.90 LMNA (0.41) LMNASIGMAR1KCNH2CYP2D6NR1I2
SCHEMBL6911992 0.90 LMNA (0.41) LMNASIGMAR1KCNH2CYP2D6NR1I2
SCHEMBL6910683 0.90 LMNA (0.41) LMNASIGMAR1KCNH2CYP2D6NR1I2
Hydrochloric Acid SCHEMBL6912979 0.90 LMNA (0.41) LMNASIGMAR1KCNH2CYP2D6NR1I2
Hydrochloric Acid SCHEMBL6916209 0.89 LMNA (0.40) LMNASIGMAR1KCNH2CYP2D6NR1I2
SCHEMBL6915496 0.87 ACHE (0.49) LMNASIGMAR1KCNH2CYP2D6NR1I2
Hydrochloric Acid SCHEMBL6914315 0.86 SIGMAR1 (0.48) LMNASIGMAR1KCNH2CYP2D6NR1I2
SCHEMBL6910631 0.81 ACHE (0.46) LMNASIGMAR1KCNH2CYP2D6NR1I2
Hydrochloric Acid SCHEMBL6911044 0.80 ACHE (0.45) LMNASIGMAR1KCNH2CYP2D6NR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1112998-B1 AMINE DERIVATIVES POLA CHEM IND INC (JP) 2004-12-08 EP disclosed
US-6586633-B1 Antifungal agents POLA CHEMICAL INDUSTRIES, INC. (JP) 2003-07-01 US disclosed
EP-1112998-A1 AMINE DERIVATIVES POLA CHEMICAL INDUSTRIES, INC. (JP) 2001-07-04 EP disclosed