SCHEMBL6911992

SCHEMBL6911992

C=C(C)c1cc(Br)cc(CN(C)Cc2ccc(C(C)(C)C)cc2)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.41
SIGMAR1 Q99720 2/20 0.41
CYP2D6 P10635 2/20 0.41
KCNH2 Q12809 2/20 0.41
NR1I2 O75469 1/20 0.41
ADRA2A P08913 1/20 0.41
ACHE P22303 1/20 0.41
SLC6A2 P23975 1/20 0.41
HTR2A P28223 1/20 0.41
SLC6A4 P31645 1/20 0.41
TMEM97 Q5BJF2 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
HIF1A Q16665 1/20 0.37
PYCR1 P32322 2/20 0.36
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6907017 0.90 LMNA (0.46) LMNASIGMAR1CYP2D6KCNH2NR1I2
SCHEMBL6910551 0.85 LMNA (0.42) LMNASIGMAR1CYP2D6KCNH2NR1I2
SCHEMBL6913929 0.84 CYP2D6 (0.50) LMNASIGMAR1CYP2D6KCNH2NR1I2
SCHEMBL6910683 0.84 LMNA (0.41) LMNASIGMAR1CYP2D6KCNH2NR1I2
SCHEMBL6914310 0.84 LMNA (0.41) LMNASIGMAR1CYP2D6KCNH2NR1I2
Hydrochloric Acid SCHEMBL6912979 0.84 LMNA (0.41) LMNASIGMAR1CYP2D6KCNH2NR1I2
Hydrochloric Acid SCHEMBL6916209 0.83 LMNA (0.40) LMNASIGMAR1CYP2D6KCNH2NR1I2
SCHEMBL6915496 0.81 ACHE (0.49) LMNASIGMAR1CYP2D6KCNH2NR1I2
Hydrochloric Acid SCHEMBL6914315 0.80 SIGMAR1 (0.48) LMNASIGMAR1CYP2D6KCNH2NR1I2
SCHEMBL6905693 0.80 CYP2D6 (0.44) LMNASIGMAR1CYP2D6KCNH2NR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1112998-B1 AMINE DERIVATIVES POLA CHEM IND INC (JP) 2004-12-08 EP disclosed
US-6586633-B1 Antifungal agents POLA CHEMICAL INDUSTRIES, INC. (JP) 2003-07-01 US disclosed
EP-1112998-A1 AMINE DERIVATIVES POLA CHEMICAL INDUSTRIES, INC. (JP) 2001-07-04 EP disclosed