SCHEMBL6909830

SCHEMBL6909830

Nc1cccc(S(=O)(=O)N2CCc3c([nH]n(Cc4ccccc4)c3=O)C2)c1

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 8/20 0.41
PKM P14618 4/20 0.40
PKLR P30613 1/20 0.40
AKR1C2 P52895 2/20 0.39
NR3C1 P04150 2/20 0.38
KDM4E B2RXH2 2/20 0.38
ALDH1A1 P00352 2/20 0.38
GAA P10253 1/20 0.38
TSHR P16473 1/20 0.38
HSD17B10 Q99714 1/20 0.38
AKR1C1 Q04828 3/20 0.38
NPSR1 Q6W5P4 1/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2356115 0.90 MEN1 (0.46) PKMNR3C1KDM4EALDH1A1TSHR
SCHEMBL14150516 0.89 NR3C1 (0.49) AKR1C3AKR1C2NR3C1KDM4EALDH1A1
SCHEMBL2357824 0.88 PKM (0.44) AKR1C3PKMPKLRAKR1C2NR3C1
SCHEMBL2354783 0.87 NR3C1 (0.51) AKR1C3PKMNR3C1ALDH1A1TSHR
SCHEMBL2347062 0.85 AKR1C3 (0.43) AKR1C3AKR1C2NR3C1KDM4EALDH1A1
SCHEMBL14150535 0.83 NR3C1 (0.47) PKMNR3C1KDM4EALDH1A1MEN1
SCHEMBL2355541 0.82 MEN1 (0.49) PKMNR3C1KDM4EALDH1A1GAA
SCHEMBL2346588 0.82 CD4 (0.51) PKMNR3C1ALDH1A1GAATSHR
SCHEMBL2348930 0.82 ALDH1A1 (0.42) KDM4EALDH1A1TSHRKMT2A
SCHEMBL2356653 0.82 LMNA (0.55) PKMPKLRNR3C1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011101805-A1 PYRAZOLO PIPERIDINE DERIVATIVES AS NADPH OXIDASE INHIBITORS GENKYOTEX SA (CH) 2011-08-25 WO disclosed