SCHEMBL6909902

SCHEMBL6909902

Clc1ccc(N2CCNCC2)s1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 7/20 0.47
HTR3E A5X5Y0 5/20 0.47
HTR3B O95264 5/20 0.47
HTR3A P46098 5/20 0.47
HTR3D Q70Z44 5/20 0.47
HTR3C Q8WXA8 5/20 0.47
SIGMAR1 Q99720 3/20 0.47
BPTF Q12830 1/20 0.46
ALDH1A1 P00352 2/20 0.44
CHRM2 P08172 1/20 0.42
CHRM4 P08173 1/20 0.42
CHRM1 P11229 1/20 0.42
CHRM3 P20309 1/20 0.42
CYP1A2 P05177 2/20 0.42
CYP3A4 P08684 2/20 0.42
HTR1A P08908 2/20 0.42
CYP2C9 P11712 2/20 0.42
HTR2A P28223 2/20 0.42
HTR2C P28335 2/20 0.42
CYP2C19 P33261 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL27237952 0.98 ADRB1 (0.46) ADRB1HTR3EHTR3BHTR3AHTR3D
SCHEMBL29999306 0.85 MAPT (0.39) ALDH1A1CYP2D6HTTMEN1HPGD
SCHEMBL81908 0.76 ADRB1 (0.47) ADRB1HTR3EHTR3BHTR3AHTR3D
SCHEMBL2247749 0.75 ALDH1A1 (0.43) ALDH1A1HTR2CTP53KMT2A
SCHEMBL1432603 0.73 AOC3 (0.40) ADRB1HTR3EHTR3BHTR3AHTR3D
SCHEMBL20080909 0.72 DRD2 (0.44) ADRB1HTR3EHTR3BHTR3AHTR3D
SCHEMBL22769076 0.72 ADRB1 (0.43) ADRB1HTR3EHTR3BHTR3AHTR3D
Hydrochloric Acid SCHEMBL28913555 0.71 DRD2 (0.42) ADRB1HTR3EHTR3BHTR3AHTR3D
SCHEMBL27237972 0.71 MAPT (0.50) ALDH1A1HTTMEN1HPGDKMT2A
SCHEMBL3851321 0.69 KDM4E (0.39) ADRB1HTR3EHTR3BHTR3AHTR3D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023011608-A1 REGULATOR CONTAINING TRICYCLIC DERIVATIVE, PREPARATION METHOD THEREFOR AND APPLICATION THEREOF 上海枢境生物科技有限公司 2023-02-09 WO disclosed
CN-113292514-B Piperazine derivative and organic photoelectric device comprising same 浙江华显光电科技有限公司 2022-11-15 CN disclosed
CN-113292514-A Piperazine derivative and organic photoelectric device comprising same 浙江华显光电科技有限公司 2021-08-24 CN disclosed
US-6825200-B1 TREATING, PROLONGING, OR EXTENDING THE ONSET OF ORGAN REJECTION IN A HUMAN DURING OR AFTER ORGAN TRANSPLANTATION IN A HUMAN FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-11-30 US disclosed
EP-1226159-A1 SUBSTITUTED DIPEPTIDES HAVING NOS INHIBITING ACTIVITY FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-07-31 EP disclosed
WO-2001032690-A1 SUBSTITUTED DIPEPTIDES HAVING NOS INHIBITING ACTIVITY FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-05-10 WO disclosed