SCHEMBL6910475

SCHEMBL6910475

COCCn1[nH]c2c(c1=O)CCN(Cc1cccc(N)c1)C2

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.41
SLC6A5 Q9Y345 1/20 0.39
MEN1 O00255 2/20 0.37
GAA P10253 1/20 0.37
ATM Q13315 1/20 0.37
DRD2 P14416 3/20 0.36
DRD4 P21917 2/20 0.36
DRD3 P35462 2/20 0.36
GNRHR P30968 1/20 0.35
ABHD6 Q9BV23 1/20 0.35
CHRM2 P08172 1/20 0.35
CHRM3 P20309 1/20 0.35
HTR1A P08908 1/20 0.35
ADRA1D P25100 1/20 0.35
ADRA1A P35348 1/20 0.35
ADRA1B P35368 1/20 0.35
ACHE P22303 1/20 0.34
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
HDAC1 Q13547 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2347548 0.88 KMT2A (0.51) KMT2ASLC6A5MEN1GAAATM
SCHEMBL2344993 0.85 CLPP (0.49) KMT2ADRD2DRD4DRD3CHRM3
SCHEMBL2349760 0.82 DRD4 (0.44) KMT2ASLC6A5MEN1GAAATM
SCHEMBL2347846 0.82 COMT (0.41)
SCHEMBL2345757 0.80 KMT2A (0.40) KMT2ASLC6A5MEN1GAAATM
SCHEMBL6911739 0.78 SLC6A5 (0.42) KMT2ASLC6A5MEN1GAAATM
SCHEMBL6910949 0.77 CHRM2 (0.42) KMT2ASLC6A5MEN1GAAATM
SCHEMBL6908510 0.76 ACHE (0.46) KMT2ASLC6A5MEN1CHRM2CHRM3
SCHEMBL2349611 0.76 MEN1 (0.48) KMT2ASLC6A5MEN1GAAATM
SCHEMBL2358094 0.76 SIGMAR1 (0.56) KMT2ASLC6A5DRD2DRD4DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011101805-A1 PYRAZOLO PIPERIDINE DERIVATIVES AS NADPH OXIDASE INHIBITORS GENKYOTEX SA (CH) 2011-08-25 WO disclosed