SCHEMBL6910600

SCHEMBL6910600

CC(=O)c1c(F)cc(C(F)(F)F)cc1C(F)(F)F

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 1/20 0.42
CES2 O00748 3/20 0.42
NOTUM Q6P988 1/20 0.37
APP P05067 1/20 0.36
MAPT P10636 1/20 0.36
GAA P10253 1/20 0.36
PDE2A O00408 1/20 0.35
MEN1 O00255 1/20 0.35
TSHR P16473 1/20 0.35
KMT2A Q03164 1/20 0.35
TRPA1 O75762 2/20 0.35
POLQ O75417 1/20 0.35
TLR7 Q9NYK1 1/20 0.34
RXRA P19793 1/20 0.34
RXRB P28702 1/20 0.34
RXRG P48443 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30628783 0.88 CES2 (0.47) KIF11CES2NOTUMMAPTMEN1
SCHEMBL423246 0.83 CES2 (0.43) CES2APPRXRARXRBRXRG
SCHEMBL30532294 0.83 CES2 (0.43) CES2APPRXRARXRBRXRG
SCHEMBL15901970 0.81 CES2 (0.42) KIF11CES2NOTUMAPPMAPT
SCHEMBL26981507 0.80 ALDH1A1 (0.42) KIF11CES2APPMAPTGAA
SCHEMBL6909178 0.79 CES2 (0.40) KIF11CES2NOTUMMAPTPOLQ
SCHEMBL18378522 0.76 CES2 (0.41) CES2NOTUMMAPT
SCHEMBL6908816 0.75 IDO1 (0.38) CES2
SCHEMBL23364827 0.74 CES2 (0.46) CES2NOTUMMAPTMEN1KMT2A
SCHEMBL16398808 0.74 CES2 (0.46) CES2APPMAPTTLR7RXRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011023667-A1 CARBOCYCLIC GLYT1 RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2011-03-03 WO disclosed