SCHEMBL6910908

SCHEMBL6910908

NCCn1[nH]c2c(c1=O)CCN(Cc1cccc(C(F)(F)F)c1)C2

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.46
ALDH1A1 P00352 1/20 0.46
GAA P10253 1/20 0.46
LMNA P02545 1/20 0.45
CLPP Q16740 2/20 0.45
BRS3 P32247 1/20 0.44
DRD2 P14416 1/20 0.43
DRD3 P35462 1/20 0.43
KCNH2 Q12809 1/20 0.43
TACR1 P25103 2/20 0.43
ADORA1 P30542 1/20 0.42
SLC6A5 Q9Y345 1/20 0.41
DAO P14920 1/20 0.40
CHRM3 P20309 1/20 0.39
TAAR1 Q96RJ0 1/20 0.39
FAAH O00519 1/20 0.39
TRPV1 Q8NER1 1/20 0.39
PARP1 P09874 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
SIGMAR1 Q99720 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2349570 0.88 CNR2 (0.44) KDM4EALDH1A1GAALMNABRS3
SCHEMBL2346409 0.81 TACR1 (0.45) KDM4EALDH1A1GAALMNACLPP
SCHEMBL6911024 0.80 BRS3 (0.44) KDM4EALDH1A1GAALMNACLPP
SCHEMBL2356534 0.76 TACR1 (0.46) KDM4EALDH1A1GAALMNACLPP
SCHEMBL2343382 0.75 UBE2M (0.41) KDM4EALDH1A1GAALMNACLPP
SCHEMBL2349473 0.74 MEN1 (0.53) GAACLPPDRD2DRD3KCNH2
SCHEMBL2439744 0.74 KDM4E (0.62) KDM4EALDH1A1GAALMNABRS3
SCHEMBL6910475 0.74 KMT2A (0.41) KDM4EALDH1A1GAADRD2DRD3
SCHEMBL2351683 0.73 MEN1 (0.53) GAACLPPDRD2DRD3KCNH2
SCHEMBL2348073 0.73 SLC6A5 (0.60) KDM4EALDH1A1GAACLPPDRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011101805-A1 PYRAZOLO PIPERIDINE DERIVATIVES AS NADPH OXIDASE INHIBITORS GENKYOTEX SA (CH) 2011-08-25 WO disclosed