SCHEMBL6911024

SCHEMBL6911024

Nc1cccc(-n2[nH]c3c(c2=O)CCN(Cc2cccc(C(F)(F)F)c2)C3)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRS3 P32247 1/20 0.44
ALDH1A1 P00352 2/20 0.43
KDM4E B2RXH2 2/20 0.43
GAA P10253 1/20 0.43
HTR1A P08908 1/20 0.43
LMNA P02545 2/20 0.43
ADORA1 P30542 1/20 0.42
TACR1 P25103 2/20 0.41
TRPV1 Q8NER1 1/20 0.41
TP53 P04637 2/20 0.40
MAPT P10636 2/20 0.40
RXFP1 Q9HBX9 1/20 0.40
DRD2 P14416 1/20 0.39
DRD3 P35462 1/20 0.39
KCNH2 Q12809 1/20 0.39
SLC6A5 Q9Y345 1/20 0.39
TSHR P16473 2/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6909785 0.93 BRS3 (0.44) BRS3ALDH1A1KDM4EGAAHTR1A
SCHEMBL6911739 0.90 SLC6A5 (0.42) GAAHTR1AADORA1DRD2SLC6A5
SCHEMBL2356534 0.86 TACR1 (0.46) BRS3ALDH1A1KDM4EGAALMNA
SCHEMBL6911686 0.85 MEN1 (0.51) GAATRPV1MAPTDRD2DRD3
SCHEMBL2343382 0.84 UBE2M (0.41) BRS3ALDH1A1KDM4EGAALMNA
SCHEMBL6910467 0.82 COMT (0.42) KDM4EDRD2KCNH2CYP3A4POLB
SCHEMBL6911338 0.81 MEN1 (0.44) ALDH1A1KDM4EGAATRPV1MAPT
SCHEMBL2355502 0.80 CLPP (0.52) GAADRD2DRD3SLC6A5CYP3A4
SCHEMBL6910908 0.80 KDM4E (0.46) BRS3ALDH1A1KDM4EGAALMNA
SCHEMBL2342836 0.80 KCNN4 (0.41) BRS3ALDH1A1KDM4EGAALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011101805-A1 PYRAZOLO PIPERIDINE DERIVATIVES AS NADPH OXIDASE INHIBITORS GENKYOTEX SA (CH) 2011-08-25 WO disclosed