SCHEMBL6915719

SCHEMBL6915719

Nc1nccc(-c2cc(C(=O)c3ccccc3)ccc2O)n1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 2/20 0.49
CDK1 P06493 8/20 0.48
CDK2 P24941 7/20 0.48
KDM4C Q9H3R0 2/20 0.48
PRKACA P17612 2/20 0.45
AURKA O14965 1/20 0.45
HSP90AA1 P07900 1/20 0.45
ADORA2A P29274 1/20 0.45
CDK5 Q00535 2/20 0.44
CDK5R1 Q15078 2/20 0.44
CCNT1 O60563 2/20 0.42
CCNB2 O95067 2/20 0.42
CCNB1 P14635 2/20 0.42
CCNA2 P20248 2/20 0.42
GSK3B P49841 2/20 0.42
CDK9 P50750 2/20 0.42
CCNA1 P78396 2/20 0.42
CCNB3 Q8WWL7 2/20 0.42
PDPK1 O15530 1/20 0.42
HTR1A P08908 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6920709 0.94 HSP90AA1 (0.49) DYRK1ACDK1CDK2KDM4CPRKACA
SCHEMBL6826600 0.93 CDK1 (0.53) DYRK1ACDK1CDK2KDM4CPRKACA
SCHEMBL7174693 0.92 PRKACA (0.47) DYRK1ACDK1CDK2KDM4CPRKACA
SCHEMBL6824620 0.91 CDK1 (0.49) DYRK1ACDK1CDK2KDM4CPRKACA
SCHEMBL6823684 0.88 CDK2 (0.47) DYRK1ACDK1CDK2KDM4CPRKACA
SCHEMBL7067140 0.84 CDK2 (0.46) DYRK1ACDK1CDK2KDM4CPRKACA
SCHEMBL6695200 0.80 KDM1A (0.49) KDM4CMEN1NPC1RAB9AKMT2A
SCHEMBL6826566 0.80 CYP2D6 (0.46) CDK1CDK2CDC7JAK2
SCHEMBL6826746 0.79 CDK1 (0.44) CDK1CDK2KDM4CPRKACACDK5
SCHEMBL6823872 0.77 CDK1 (0.54) DYRK1ACDK1CDK2JAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004080979-A1 NOVEL 3-(2-AMINO-4-PYRIMIDINYL)-4-HYDROXYPHENYL KETONE DERIVATIVES LG LIFE SCIENCES LTD. (KR) 2004-09-23 WO disclosed