SCHEMBL7174693

SCHEMBL7174693

Nc1nccc(-c2cc(C(=O)c3cccc(-c4ccccc4)c3)ccc2O)n1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKACA P17612 2/20 0.47
ADORA2A P29274 2/20 0.47
AURKA O14965 1/20 0.47
HSP90AA1 P07900 1/20 0.47
CDK1 P06493 7/20 0.45
CDK2 P24941 7/20 0.45
DYRK1A Q13627 2/20 0.45
GSK3B P49841 3/20 0.44
CCNT1 O60563 2/20 0.44
CCNB2 O95067 2/20 0.44
CCNB1 P14635 2/20 0.44
CCNA2 P20248 2/20 0.44
CDK9 P50750 2/20 0.44
CCNA1 P78396 2/20 0.44
CCNB3 Q8WWL7 2/20 0.44
PDPK1 O15530 1/20 0.44
HTR1A P08908 1/20 0.44
PRKACG P22612 1/20 0.44
PRKACB P22694 1/20 0.44
HTR2B P41595 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6920709 0.93 HSP90AA1 (0.49) PRKACAADORA2AAURKAHSP90AA1CDK1
SCHEMBL6915719 0.92 DYRK1A (0.49) PRKACAADORA2AAURKAHSP90AA1CDK1
SCHEMBL6826600 0.88 CDK1 (0.53) PRKACAADORA2AAURKAHSP90AA1CDK1
SCHEMBL6824620 0.83 CDK1 (0.49) PRKACACDK1CDK2DYRK1AGSK3B
SCHEMBL7067140 0.81 CDK2 (0.46) PRKACACDK1CDK2DYRK1AGSK3B
SCHEMBL6823684 0.81 CDK2 (0.47) PRKACACDK1CDK2DYRK1AGSK3B
SCHEMBL6826566 0.77 CYP2D6 (0.46) CDK1CDK2CDC7JAK2CYP2C9
SCHEMBL6642333 0.76 CDK2 (0.53) PRKACAADORA2AAURKAHSP90AA1CDK1
SCHEMBL6638867 0.75 CDK1 (0.58) PRKACAADORA2AAURKAHSP90AA1CDK1
SCHEMBL4202167 0.75 HSP90AA1 (0.76) PRKACAADORA2AAURKAHSP90AA1CDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004080979-A1 NOVEL 3-(2-AMINO-4-PYRIMIDINYL)-4-HYDROXYPHENYL KETONE DERIVATIVES LG LIFE SCIENCES LTD. (KR) 2004-09-23 WO disclosed