SCHEMBL6823684

SCHEMBL6823684

Nc1nccc(-c2cc(C(=O)c3ccc(Cl)cc3)ccc2O)n1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 9/20 0.47
CDK1 P06493 8/20 0.47
GSK3B P49841 3/20 0.44
DYRK1A Q13627 2/20 0.44
MAP3K14 Q99558 1/20 0.44
AGPAT2 O15120 1/20 0.44
CDK5 Q00535 3/20 0.43
CDK5R1 Q15078 1/20 0.43
JAK2 O60674 5/20 0.42
CDK9 P50750 4/20 0.42
CDC7 O00311 3/20 0.42
CSNK1A1 P48729 3/20 0.42
CSNK1D P48730 3/20 0.42
CSNK2A1 P68400 3/20 0.42
MAPK1 P28482 3/20 0.42
CCNT1 O60563 2/20 0.42
MAP4K4 O95819 2/20 0.42
PLK4 O00444 2/20 0.42
MAPK13 O15264 2/20 0.42
DAPK3 O43293 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6826600 0.92 CDK1 (0.53) CDK2CDK1GSK3BDYRK1ACDK5
SCHEMBL6824620 0.90 CDK1 (0.49) CDK2CDK1GSK3BDYRK1ACDK5
SCHEMBL6915719 0.88 DYRK1A (0.49) CDK2CDK1GSK3BDYRK1ACDK5
SCHEMBL6920709 0.85 HSP90AA1 (0.49) CDK2CDK1GSK3BDYRK1ACDK5
SCHEMBL7174693 0.81 PRKACA (0.47) CDK2CDK1GSK3BDYRK1ACDK5
SCHEMBL7067140 0.80 CDK2 (0.46) CDK2CDK1GSK3BDYRK1ACDK5
SCHEMBL6826746 0.78 CDK1 (0.44) CDK2CDK1GSK3BCDK5CDK5R1
SCHEMBL6922661 0.78 CDK2 (0.51) CDK2CDK1GSK3BDYRK1AMAP3K14
SCHEMBL5803933 0.74 CDK1 (0.58) CDK2CDK1GSK3BDYRK1AMAP3K14
SCHEMBL6826566 0.74 CYP2D6 (0.46) CDK2CDK1JAK2CDC7JAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004080979-A1 NOVEL 3-(2-AMINO-4-PYRIMIDINYL)-4-HYDROXYPHENYL KETONE DERIVATIVES LG LIFE SCIENCES LTD. (KR) 2004-09-23 WO disclosed