SCHEMBL6918826

SCHEMBL6918826

O=C(O)C[C@@H]1CC[C@@H](N(Cc2cccc(F)c2)CC2CCCC2)[C@H](c2ccc(CF)cc2)C1

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PKM P14618 2/20 0.39
DGAT1 O75907 2/20 0.36
SLC6A2 P23975 1/20 0.35
SLC6A3 Q01959 1/20 0.35
OPRM1 P35372 7/20 0.35
OPRD1 P41143 2/20 0.35
STAT3 P40763 2/20 0.34
IDH1 O75874 1/20 0.33
KDM1A O60341 2/20 0.32
SIGMAR1 Q99720 1/20 0.32
TSPO P30536 1/20 0.32
MAOA P21397 1/20 0.32
MAOB P27338 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2315428 0.90 PKM (0.38) PKMDGAT1SLC6A2SLC6A3OPRM1
SCHEMBL6917782 0.80 SIGMAR1 (0.45) DGAT1SLC6A2SIGMAR1
SCHEMBL2315414 0.80 MDM2 (0.37) DGAT1
SCHEMBL2318519 0.80 SIGMAR1 (0.37) PKMSLC6A2SIGMAR1MAOA
SCHEMBL6918642 0.80 MAOA (0.39) SLC6A2KDM1AMAOAMAOB
SCHEMBL10032827 0.76 GPR88 (0.42) KDM1ASIGMAR1MAOAMAOB
SCHEMBL2316326 0.76 PSEN1 (0.42) SLC6A2MAOA
SCHEMBL6916644 0.74 MDM2 (0.40) OPRM1KDM1AMAOAMAOB
SCHEMBL2315082 0.74 SLC6A2 (0.38) PKMDGAT1SLC6A2SLC6A3MAOA
SCHEMBL2317127 0.74 PSEN1 (0.41) DGAT1SIGMAR1MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011092611-A1 AMINOCYCLOHEXANES AND AMINOTETRAHYDROPYRANS AND RELATED COMPOUNDS AS GAMMA-SECRETASE MODULATORS PFIZER INC. (US) 2011-08-04 WO disclosed