SCHEMBL6919652

SCHEMBL6919652

COc1nc(OC)nc(N2CCN(c3ncc(C(=O)N4CCCC4)cc3Cl)CC2)n1

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
P2RY12 Q9H244 9/20 0.45
CXCR3 P49682 2/20 0.45
GRM5 P41594 2/20 0.44
HSD17B10 Q99714 1/20 0.44
TRPV1 Q8NER1 1/20 0.42
KDM4E B2RXH2 1/20 0.41
GBA1 P04062 1/20 0.41
LRRK2 Q5S007 2/20 0.41
MEN1 O00255 1/20 0.41
HTT P42858 1/20 0.41
RECQL P46063 1/20 0.41
KMT2A Q03164 1/20 0.41
ATM Q13315 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6826032 0.79 P2RY12 (0.49) P2RY12CXCR3GRM5
SCHEMBL6916055 0.78 HSD11B1 (0.45) P2RY12CXCR3GRM5HSD17B10
SCHEMBL13648884 0.75 CXCR3 (0.55) CXCR3LRRK2
Hydrochloric Acid SCHEMBL3976856 0.74 CXCR3 (0.54) CXCR3LRRK2
SCHEMBL6919706 0.73 CYP2C9 (0.45) P2RY12CXCR3GRM5KDM4EMEN1
SCHEMBL6826225 0.73 HPGD (0.49) CXCR3MEN1KMT2A
SCHEMBL6820189 0.72 CXCR3 (0.44) P2RY12CXCR3GRM5KDM4E
SCHEMBL6917988 0.72 CCR4 (0.44) P2RY12CXCR3GRM5
SCHEMBL6823744 0.72 KMT2A (0.48) P2RY12CXCR3GRM5HSD17B10KDM4E
SCHEMBL6820208 0.72 CXCR3 (0.43) P2RY12CXCR3GRM5KDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004074287-A1 NOVEL COMPOUNDS ASTRAZENECA AB (SE) 2004-09-02 WO claimed
WO-2004074287-A1 NOVEL COMPOUNDS ASTRAZENECA AB (SE) 2004-09-02 WO disclosed