SCHEMBL6921782

SCHEMBL6921782

O=c1c2ccc(-c3cccc(F)c3)cc2nc2n1CC1CCC(C2)N1

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GSK3A P49840 1/20 0.36
GSK3B P49841 1/20 0.36
PAX8 Q06710 1/20 0.36
TNKS2 Q9H2K2 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CACNA2D1 P54289 1/20 0.34
NT5E P21589 1/20 0.34
CTSD P07339 2/20 0.34
BCL2A1 Q16548 1/20 0.33
IDO1 P14902 1/20 0.33
BACE1 P56817 1/20 0.33
MAP4K4 O95819 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12041886 0.85 GRM5 (0.39)
SCHEMBL12059022 0.83 GRM2 (0.39) TNKS2CYP1A2CYP3A4NT5ECTSD
SCHEMBL12059074 0.79 LMNA (0.38) TNKS2BCL2A1BACE1
SCHEMBL6921125 0.79 RAB9A (0.40) GSK3AGSK3BCYP1A2CYP3A4
SCHEMBL12059019 0.78 CTSD (0.36) TNKS2CTSDBCL2A1BACE1MAP4K4
SCHEMBL12059079 0.78 BCL2A1 (0.38) CYP1A2CYP3A4CTSDBCL2A1
SCHEMBL6922345 0.77 HTR1A (0.41) TNKS2MAP4K4
SCHEMBL6920638 0.76 RAB9A (0.38) GSK3AGSK3BCYP1A2CYP3A4
SCHEMBL6920625 0.76 APOBEC3A (0.37) GSK3AGSK3BTNKS2CYP1A2CYP3A4
SCHEMBL12059544 0.76 GRM2 (0.37) CYP1A2CYP3A4CTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011075699-A2 COMPOUNDS FOR TREATING DISORDERS MEDIATED BY METABOTROPIC GLUTAMATE RECEPTOR 5, AND METHODS OF USE THEREOF SUNOVION PHARMACEUTICALS INC. (US) 2011-06-23 WO disclosed